SCHEMBL4747267

SCHEMBL4747267

CC[C@@](Cc1ccc2nc(-c3c(Cl)cccc3Cl)ccc2c1)(NC(=O)OC(C)(C)C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.47
ITGAV P06756 1/20 0.47
ABL1 P00519 1/20 0.37
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
AAK1 Q2M2I8 8/20 0.33
LCK P06239 2/20 0.33
ACACB O00763 1/20 0.33
ACACA Q13085 1/20 0.33
ACSS2 Q9NR19 1/20 0.33
DGAT1 O75907 1/20 0.33
P2RX7 Q99572 1/20 0.33
CTSL P07711 1/20 0.33
PPARG P37231 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32
PTPN1 P18031 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1030228 0.88 ITGB1 (0.49) ITGB1ITGAVABL1CTSBCTSS
SCHEMBL3318595 0.80 ITGB1 (0.71) ITGB1ITGAVCTSBCTSSCTSK
SCHEMBL4626858 0.80 ITGB1 (0.71) ITGB1ITGAVCTSBCTSSCTSK
SCHEMBL3315439 0.80 ITGB1 (0.71) ITGB1ITGAVCTSBCTSSCTSK
SCHEMBL4747262 0.78 ITGB1 (0.58) ITGB1ITGAVCTSBCTSSCTSK
SCHEMBL4750015 0.77 ITGB1 (0.53) ITGB1ITGAVABL1
SCHEMBL4626504 0.77 ITGB1 (0.53) ITGB1ITGAVABL1
SCHEMBL1030225 0.77 ITGB1 (0.59) ITGB1ITGAVCTSBCTSSCTSK
SCHEMBL3320795 0.77 ITGB1 (0.59) ITGB1ITGAVCTSBCTSSCTSK
SCHEMBL4627521 0.77 ITGB1 (0.59) ITGB1ITGAVCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008138592-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-11-20 WO disclosed
WO-2008125215-A1 BICYCLIC AND HETEROBICYCLIC DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES UCB PHARMA, S.A. (BE) 2008-10-23 WO disclosed