SCHEMBL4748772

SCHEMBL4748772

O=C(C=Cc1ccc(Nc2ccnc3cc(Cl)ccc23)cc1)c1ccc(F)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.56
MAPT P10636 2/20 0.56
ATM Q13315 1/20 0.56
CYP2D6 P10635 8/20 0.51
CYP1A2 P05177 7/20 0.51
TNFRSF1A P19438 1/20 0.48
PTGS2 P35354 2/20 0.48
MET P08581 1/20 0.48
CYP2C8 P10632 5/20 0.47
CYP2C19 P33261 5/20 0.47
KCNH2 Q12809 4/20 0.47
CYP2C9 P11712 3/20 0.47
CYP3A4 P08684 2/20 0.46
MAPKAPK2 P49137 1/20 0.46
ABCB11 O95342 1/20 0.46
APP P05067 1/20 0.46
CHRM2 P08172 1/20 0.46
HTR1A P08908 1/20 0.46
CHRM1 P11229 1/20 0.46
DRD2 P14416 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4748776 1.00 GAA (0.56) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL14024383 1.00 GAA (0.56) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL14024382 0.94 MAPT (0.60) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL4748929 0.94 MAPT (0.60) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL4748932 0.94 MAPT (0.60) GAAMAPTATMCYP2D6CYP1A2
Citric Acid SCHEMBL25202377 0.90 GAA (0.46) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL14024394 0.85 MAPT (0.59) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL4752430 0.85 MAPT (0.59) GAAMAPTATMCYP2D6CYP1A2
SCHEMBL4752428 0.84 CYP2D6 (0.58) GAAMAPTATMCYP2D6CYP1A2
Citric Acid SCHEMBL25210605 0.84 GAA (0.48) GAAMAPTATMCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135886-A2 QUINOLINE DERIVATIVES FOR USE IN THE INHIBITION OF THE GROWTH OF TUMOUR CELLS UNIVERSITY OF PRETORIA (ZA) 2008-11-13 WO disclosed