SCHEMBL4748932

SCHEMBL4748932

O=C(C=Cc1ccc(Cl)cc1)c1ccc(Nc2ccnc3cc(Cl)ccc23)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.60
GAA P10253 2/20 0.60
ATM Q13315 1/20 0.60
CYP2D6 P10635 6/20 0.54
CYP1A2 P05177 5/20 0.54
MAPKAPK2 P49137 1/20 0.52
TDP1 Q9NUW8 2/20 0.51
KMT2A Q03164 1/20 0.51
EGFR P00533 2/20 0.48
KCNH2 Q12809 3/20 0.48
ABCB11 O95342 1/20 0.48
APP P05067 1/20 0.48
CHRM2 P08172 1/20 0.48
HTR1A P08908 1/20 0.48
CHRM1 P11229 1/20 0.48
DRD2 P14416 1/20 0.48
ADRA2C P18825 1/20 0.48
SLC6A2 P23975 1/20 0.48
PTGS2 P35354 1/20 0.48
OPRM1 P35372 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4748929 1.00 MAPT (0.60) MAPTGAAATMCYP2D6CYP1A2
SCHEMBL14024382 1.00 MAPT (0.60) MAPTGAAATMCYP2D6CYP1A2
SCHEMBL4748772 0.94 GAA (0.56) MAPTGAAATMCYP2D6CYP1A2
SCHEMBL14024383 0.94 GAA (0.56) MAPTGAAATMCYP2D6CYP1A2
SCHEMBL4748776 0.94 GAA (0.56) MAPTGAAATMCYP2D6CYP1A2
Citric Acid SCHEMBL25210605 0.89 GAA (0.48) MAPTGAAATMCYP2D6CYP1A2
SCHEMBL4748784 0.89 CYP2D6 (0.52) MAPTGAAATMCYP2D6CYP1A2
SCHEMBL14024396 0.89 CYP2D6 (0.52) MAPTGAAATMCYP2D6CYP1A2
SCHEMBL4748788 0.89 CYP2D6 (0.52) MAPTGAAATMCYP2D6CYP1A2
SCHEMBL4752430 0.88 MAPT (0.59) MAPTGAAATMCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135886-A2 QUINOLINE DERIVATIVES FOR USE IN THE INHIBITION OF THE GROWTH OF TUMOUR CELLS UNIVERSITY OF PRETORIA (ZA) 2008-11-13 WO disclosed