SCHEMBL4750460

SCHEMBL4750460

O=C(N[C@@H]1COc2cccc(NCCN3CCCC3)c2C1)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 15/20 0.65
SCN5A Q14524 11/20 0.65
KCNH2 Q12809 11/20 0.65
HTR2A P28223 3/20 0.43
DRD3 P35462 2/20 0.43
EPHX2 P34913 1/20 0.43
MCHR1 Q99705 1/20 0.42
DRD4 P21917 1/20 0.41
DRD2 P14416 1/20 0.41
SLC6A3 Q01959 1/20 0.40
GHSR Q92847 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750039 0.85 SCN9A (0.66) SCN9ASCN5AKCNH2HTR2ADRD3
SCHEMBL4750025 0.84 SCN9A (0.65) SCN9ASCN5AKCNH2HTR2ADRD3
SCHEMBL4842078 0.79 SCN9A (1.00) SCN9ASCN5AKCNH2HTR2ADRD3
SCHEMBL4842065 0.79 SCN9A (1.00) SCN9ASCN5AKCNH2HTR2ADRD3
SCHEMBL4749982 0.77 SCN9A (0.77) SCN9ASCN5AKCNH2HTR2ADRD3
SCHEMBL4747089 0.76 SCN9A (0.73) SCN9ASCN5AKCNH2HTR2ADRD3
SCHEMBL4747549 0.76 SCN9A (0.69) SCN9ASCN5AKCNH2HTR2ADRD3
SCHEMBL4747610 0.75 SCN9A (0.52) SCN9ASCN5AKCNH2SLC6A3GHSR
SCHEMBL839807 0.74 SCN9A (1.00) SCN9ASCN5AKCNH2SLC6A3GHSR
SCHEMBL840903 0.73 SCN9A (1.00) SCN9ASCN5AKCNH2SLC6A3GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130319-A2 NOVEL N-TETRAHYDRONAPHTALENE OR N-CHROMANE CARBOXAMIDE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed