SCHEMBL4751259

SCHEMBL4751259

COCCNc1nc2cc(Cl)ccc2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
MCHR1 Q99705 1/20 0.46
ALDH1A1 P00352 2/20 0.44
NPC1 O15118 3/20 0.43
POLB P06746 2/20 0.43
KLF5 Q13887 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
KCNH2 Q12809 1/20 0.43
HRH4 Q9H3N8 2/20 0.43
BCHE P06276 1/20 0.43
TRPC3 Q13507 1/20 0.43
TRPC4 Q9UBN4 1/20 0.43
TRPC5 Q9UL62 1/20 0.43
PYGL P06737 1/20 0.41
EIF2AK2 P19525 1/20 0.41
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5100530 0.81 CYP1A2 (0.57) RAB9ACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL5096961 0.81 RAB9A (0.52) RAB9ACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL13049808 0.80 BCHE (0.66) RAB9AALDH1A1NPC1POLBTDP1
SCHEMBL5103712 0.76 CYP1A2 (0.51) RAB9ACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL4151151 0.76 HRH4 (0.47) RAB9ACYP1A2CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL28371344 0.74 RAB9A (0.48) RAB9ACYP1A2CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL4159988 0.74 RAB9A (0.48) RAB9ACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL13733061 0.74 SMN1; SMN2 (0.56) RAB9ACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL11171719 0.73 NPC1 (0.55) RAB9ACYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL16342365 0.72 RAB9A (0.45) RAB9ACYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135526-A1 CARBOXYLIC ACID AMIDES AS FACTOR XA INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-13 WO disclosed