SCHEMBL4751365

SCHEMBL4751365

COc1cc(I)c(CCO)cc1OC(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.43
HTR2C P28335 3/20 0.43
HTR2B P41595 3/20 0.43
HTR1A P08908 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
PMP22 Q01453 2/20 0.42
LMNA P02545 1/20 0.42
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
HMGCR P04035 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
ACHE P22303 1/20 0.35
TAAR1 Q96RJ0 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750269 0.91 HTR2A (0.41) HTR2AHTR2CHTR2BHTR1ACYP1A2
SCHEMBL25143222 0.88 MTNR1A (0.45) HTR2AHTR2CHTR2BHTR1ACYP1A2
SCHEMBL4750246 0.84 SMN1; SMN2 (0.45) HTR2AHTR2CLMNATAAR1
SCHEMBL5355957 0.74 PDE4A (0.46) HTR2AHTR2CLMNAMTNR1AMTNR1B
SCHEMBL4982275 0.74 PDE4A (0.57) HTR2AHTR2CHTR2BHTR1ACYP1A2
SCHEMBL661243 0.72 MGAM (0.42) HTR2AHTR2CHTR2BHTR1ACYP1A2
SCHEMBL5350260 0.72 HTR2A (0.43) HTR2AHTR2CLMNAMTNR1AMTNR1B
SCHEMBL3391657 0.72 HTR2A (0.52) HTR2AHTR2CHTR2BHTR1ACYP1A2
SCHEMBL21798808 0.71 TAAR1 (0.52) HTR2AHTR2CCYP3A4HMGCRPDE4A
SCHEMBL4748125 0.71 STAT3 (0.51) CYP1A2CYP3A4CYP2D6PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008124878-A1 NON-STEROIDAL COMPOUNDS CRYPTOPHARMA PTY LTD (AU) 2008-10-23 WO disclosed