SCHEMBL4751987

SCHEMBL4751987

C[C@@H](OC(=O)N1CCN(C(=O)O[C@H](C)n2cc(C3CC3)nn2)CC1)n1cc(C2CC2)nn1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.43
ATM Q13315 1/20 0.43
CYP19A1 P11511 2/20 0.37
MGLL Q99685 2/20 0.34
EPHX2 P34913 1/20 0.33
CACNA1C Q13936 1/20 0.33
GPR88 Q9GZN0 1/20 0.33
HRH3 Q9Y5N1 5/20 0.33
GPR119 Q8TDV5 4/20 0.33
PLA2G7 Q13093 1/20 0.33
ABHD6 Q9BV23 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
KDM1A O60341 1/20 0.32
GRIN2B Q13224 1/20 0.32
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751949 0.78 HTT (0.42) HTTATMMGLLHRH3GPR119
SCHEMBL12719014 0.73 CYP19A1 (0.40) HTTATMCYP19A1EPHX2CACNA1C
SCHEMBL18734148 0.72 CYP19A1 (0.49) CYP19A1GPR88
SCHEMBL31208153 0.71 HTT (0.53) HTTATMGPR119IRAK4MAPK1
SCHEMBL12719013 0.70 CYP19A1 (0.40) HTTATMCYP19A1EPHX2CACNA1C
SCHEMBL30896970 0.69 CA12 (0.45) HTTATMCYP19A1EPHX2CACNA1C
SCHEMBL4749714 0.69 HTT (0.36) HTTATMMGLLHRH3PLA2G7
SCHEMBL24438094 0.68 CYP19A1 (0.46) HTTATMCYP19A1EPHX2CACNA1C
SCHEMBL12172122 0.68 CYP19A1 (0.56) HTTATMCYP19A1GPR88HRH3
SCHEMBL24482326 0.67 CYP19A1 (0.44) HTTATMCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed