SCHEMBL4751949

SCHEMBL4751949

CC(=O)c1cn([C@@H](C)OC(=O)N2CCN(C(=O)O[C@H](C)n3cc(C(C)=O)nn3)CC2)nn1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.42
ATM Q13315 1/20 0.42
KDM1A O60341 1/20 0.33
GPR119 Q8TDV5 4/20 0.33
MAPK1 P28482 1/20 0.32
KMT2A Q03164 4/20 0.32
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 3/20 0.31
NPSR1 Q6W5P4 1/20 0.31
MGLL Q99685 2/20 0.30
FAAH O00519 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751987 0.78 HTT (0.43) HTTATMKDM1AGPR119MAPK1
SCHEMBL14262405 0.74 ACHE (0.36) ALDH1A1SMN1; SMN2NPSR1
SCHEMBL4749714 0.71 HTT (0.36) HTTATMKDM1AKMT2AL3MBTL1
SCHEMBL4753615 0.67 HDAC8 (0.41) HTTKMT2ASMN1; SMN2MEN1MGLL
SCHEMBL22021946 0.66 ACHE (0.35) ALDH1A1SMN1; SMN2NPSR1
SCHEMBL4303680 0.64 HSD17B10 (0.47) HTTALDH1A1MGLLFAAH
SCHEMBL4297220 0.64 MGLL (0.45) MAPK1KMT2AALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL27979621 0.62
SCHEMBL26317513 0.62 TSHR (0.43) HTTKDM1AGPR119ALDH1A1SMN1; SMN2
SCHEMBL3404701 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed