SCHEMBL4754891

SCHEMBL4754891

CC[C@@H]1CN(c2ncccn2)CCN1C(=O)c1ccc(-c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 18/20 0.63
SMO Q99835 1/20 0.46
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
NAMPT P43490 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4754888 1.00 SLC6A7 (0.63) SLC6A7SMOALDH1A1TSHRNAMPT
SCHEMBL3575473 0.89 SLC6A7 (0.60) SLC6A7SMOALDH1A1TSHR
SCHEMBL3575476 0.89 SLC6A7 (0.60) SLC6A7SMOALDH1A1TSHR
SCHEMBL3585161 0.87 SLC6A7 (0.60) SLC6A7SMOALDH1A1TSHR
SCHEMBL3585156 0.87 SLC6A7 (0.60) SLC6A7SMOALDH1A1TSHR
SCHEMBL3579344 0.86 SLC6A7 (0.74) SLC6A7SMOALDH1A1TSHR
SCHEMBL3579341 0.86 SLC6A7 (0.74) SLC6A7SMOALDH1A1TSHR
SCHEMBL3580071 0.86 SLC6A7 (0.74) SLC6A7SMOALDH1A1TSHR
SCHEMBL3585370 0.84 SLC6A7 (0.63) SLC6A7SMOALDH1A1TSHRNAMPT
SCHEMBL3585367 0.84 SLC6A7 (0.63) SLC6A7SMOALDH1A1TSHRNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893212-A2 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE Lexicon Pharmaceuticals, Inc. (US) 2008-03-05 EP claimed
WO-2006124748-A2 MULTICYCLIC COMPOUNDS AND METHODS OF THEIR USE LEXICON GENETICS INCORPORATED (US) 2006-11-23 WO claimed