SCHEMBL4755038

SCHEMBL4755038

Cc1nc2c(NC3CCOc4ccccc43)cc(N3CCC3=O)cc2n1C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 5/20 0.37
MAPK1 P28482 2/20 0.36
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
NTRK1 P04629 1/20 0.34
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
LRRK2 Q5S007 1/20 0.32
APOBEC3A P31941 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
CCR6 P51684 1/20 0.32
PIK3CA P42336 1/20 0.32
PFKFB3 Q16875 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755613 0.95 TRPV1 (0.36) TRPV1MAPK1CYP3A4CYP2C9CNR1
SCHEMBL13983104 0.90 TRPV1 (0.38) TRPV1MAPK1CNR2NTRK1
SCHEMBL13983099 0.85 TRPV1 (0.37) TRPV1CNR2NTRK1
SCHEMBL13983135 0.84 TRPV1 (0.37) TRPV1CYP3A4CYP2C9CNR2NTRK1
SCHEMBL13983271 0.83
SCHEMBL4755426 0.81 MAPK1 (0.36) TRPV1MAPK1CYP3A4CYP2C9CNR1
SCHEMBL13983272 0.78 TP53 (0.33)
SCHEMBL13983280 0.77 BRD9 (0.33) CYP3A4CYP2C9PIK3CA
SCHEMBL13983521 0.77 SLC9A3 (0.34) TRPV1MAPK1PIK3CA
SCHEMBL13983267 0.72 TRPV1 (0.38) TRPV1MAPK1CNR2NTRK1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151927-A2 6-N-SUBSTITUTED BENZ IMIDAZOLE DERIVATIVES AS ACID PUMP ANTAGONISTS NYCOMED GMBH (DE) 2008-12-18 WO disclosed