SCHEMBL4755309

SCHEMBL4755309

CONC(=O)C#Cc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.58
RAB9A P51151 5/20 0.58
MEN1 O00255 1/20 0.58
POLB P06746 1/20 0.58
KMT2A Q03164 1/20 0.58
NLRP3 Q96P20 1/20 0.58
NPSR1 Q6W5P4 1/20 0.50
GFER P55789 1/20 0.46
VCP P55072 3/20 0.46
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HTT P42858 1/20 0.42
MTOR P42345 1/20 0.41
HSP90AA1 P07900 1/20 0.41
AGTR1 P30556 1/20 0.41
PAX8 Q06710 1/20 0.41
TLR9 Q9NR96 1/20 0.41
UTS2R Q9UKP6 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4554708 0.79 NPSR1 (0.55) NPC1RAB9AMEN1POLBKMT2A
SCHEMBL124863 0.79 NPSR1 (0.55) NPC1RAB9AMEN1POLBKMT2A
SCHEMBL10254937 0.78 NPC1 (0.50) NPC1RAB9AMEN1POLBKMT2A
SCHEMBL7746477 0.76 NPC1 (0.49) NPC1RAB9AMEN1POLBKMT2A
SCHEMBL12426069 0.76 NPC1 (0.56) NPC1RAB9AMEN1POLBKMT2A
SCHEMBL19823669 0.76 NPC1 (0.54) NPC1RAB9AMEN1POLBKMT2A
SCHEMBL16071071 0.76 NPC1 (0.51) NPC1RAB9AMEN1POLBKMT2A
SCHEMBL7636834 0.76 NPSR1 (0.52) NPC1RAB9AMEN1POLBKMT2A
SCHEMBL6361487 0.75 PTGES (0.50) NPC1RAB9AMEN1POLBKMT2A
SCHEMBL15600987 0.74 UTS2R (0.50) NPC1RAB9AMEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968958-A1 SUBSTITUTED THIAZOLES AND THEIR USE FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2008-09-17 EP disclosed
WO-2007079961-A1 SUBSTITUTED THIAZOLES AND THEIR USE FOR PRODUCING DRUGS Grünenthal GmbH (DE) 2007-07-19 WO disclosed