SCHEMBL4756410

SCHEMBL4756410

FC1CCCc2ccccc2C1F

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.50
ADRA2A P08913 2/20 0.41
ADRA1A P35348 2/20 0.41
CYP2D6 P10635 2/20 0.41
LMNA P02545 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1B P35368 1/20 0.41
HTR1A P08908 1/20 0.41
OPRM1 P35372 1/20 0.41
HTT P42858 1/20 0.41
TSHR P16473 1/20 0.41
ALDH1A1 P00352 2/20 0.41
CHRNA7 P36544 1/20 0.41
MEN1 O00255 1/20 0.41
BLM P54132 1/20 0.41
KMT2A Q03164 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
PDPK1 O15530 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6667045 0.88 IDO1 (0.47) IDO1PDPK1
SCHEMBL30056716 0.79 IDO1 (0.53) IDO1ADRA2AADRA1ACYP2D6LMNA
SCHEMBL4248158 0.79 IDO1 (0.53) IDO1ADRA2AADRA1ACYP2D6LMNA
SCHEMBL59025 0.75 IDO1 (0.53) IDO1ADRA2AADRA1ACYP2D6LMNA
SCHEMBL10729425 0.75 IDO1 (0.53) IDO1ADRA2AADRA1ACYP2D6LMNA
SCHEMBL29357487 0.74 IDO1 (0.57) IDO1ADRA2AADRA1ACYP2D6LMNA
SCHEMBL145977 0.74 IDO1 (0.57) IDO1ADRA2AADRA1ACYP2D6LMNA
SCHEMBL16242534 0.74 MAOB (0.47)
SCHEMBL15340730 0.73 IDO1 (0.44) IDO1ALDH1A1MEN1KMT2APDPK1
SCHEMBL13082165 0.72 IDO1 (0.55) IDO1ADRA2AADRA1ACYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1976843-A2 CARBOCYCLIC AND HETEROCYCLIC ARYLSULFONES AS GAMMA SECRETASE INHIBITORS SCHERING CORPORATION (US) 2008-10-08 EP disclosed
WO-2007084595-A2 CARBOCYCLIC AND HETEROCYCLIC ARYLSULFONES AS GAMMA SECRETASE INHIBITORS SCHERING CORPORATION (US) 2007-07-26 WO disclosed