SCHEMBL4759638

SCHEMBL4759638

c1ccc2cc(CCCc3ccc(NC4=NCCN4)cc3)ccc2c1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 12/20 0.58
ADRA2B P18089 11/20 0.58
ADRA2C P18825 11/20 0.58
PTGIR P43119 4/20 0.52
CYP2D6 P10635 1/20 0.51
NFKB1 P19838 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
GPR65 Q8IYL9 1/20 0.49
AOC3 Q16853 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4759817 0.81 ADRA2A (0.54) ADRA2AADRA2BADRA2CPTGIRCYP2D6
SCHEMBL13017196 0.81 ADRA2A (0.81) ADRA2AADRA2BADRA2CPTGIRGPR65
Hydrochloric Acid SCHEMBL6161690 0.80 ADRA2A (0.53) ADRA2AADRA2BADRA2CPTGIRGPR65
SCHEMBL7081326 0.80 PTGIR (0.55) ADRA2AADRA2BADRA2CPTGIRGPR65
SCHEMBL5803363 0.78 PTGIR (0.77) ADRA2AADRA2BADRA2CPTGIR
SCHEMBL4743095 0.78 ADRA2A (0.66) ADRA2AADRA2BADRA2CPTGIRGPR65
SCHEMBL13063330 0.76 CYP2D6 (0.58) ADRA2AADRA2BADRA2CPTGIRCYP2D6
SCHEMBL13017193 0.76 ADRA2A (0.88) ADRA2AADRA2BADRA2CPTGIRCYP2D6
SCHEMBL13062961 0.76 ADRA2A (0.72) ADRA2AADRA2BADRA2CPTGIRGPR65
Hydrochloric Acid SCHEMBL4689790 0.75 ADRA2A (0.62) ADRA2AADRA2BADRA2CPTGIRGPR65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981498-A2 USE OF 2-IMIDAZOLES FOR THE TREATMENT OF CNS DISORDERS F. Hoffmann-la Roche AG (CH) 2008-10-22 EP disclosed
WO-2007090720-A2 USE OF 2-IMIDAZOLES FOR THE TREATMENT OF CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2007-08-16 WO disclosed