SCHEMBL4766874

SCHEMBL4766874

NC(=O)c1ccccc1NC(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.73

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 12/20 0.73
PTGS1 P23219 2/20 0.71
GAA P10253 1/20 0.67
ALDH1A1 P00352 1/20 0.64
LMNA P02545 1/20 0.62
KCNK3 O14649 1/20 0.59
P2RX1 P51575 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30932523 1.00 RXFP1 (0.73) RXFP1PTGS1GAAALDH1A1LMNA
SCHEMBL29085612 0.89 RXFP1 (0.67) RXFP1PTGS1GAAALDH1A1P2RX1
SCHEMBL15775396 0.86 PTGS1 (0.68) RXFP1PTGS1
SCHEMBL6720875 0.85 MEN1 (0.73) ALDH1A1LMNA
SCHEMBL15530200 0.84 RXFP1 (1.00) RXFP1
SCHEMBL30112566 0.82 RXFP1 (0.79) RXFP1
SCHEMBL28473857 0.82 RXFP1 (0.79) RXFP1
SCHEMBL28633823 0.82 PTGS1 (0.72) RXFP1PTGS1GAAALDH1A1LMNA
SCHEMBL11868617 0.82 PTGS1 (0.72) RXFP1PTGS1GAAALDH1A1LMNA
SCHEMBL30136206 0.82 PTGS1 (0.72) RXFP1PTGS1GAAALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108779078-A New inhibitor and probe of kinases and application thereof 北京大学深圳研究生院 2018-11-09 CN disclosed
EP-1928844-A2 BIS-ARYL AMIDE COMPOUNDS AND METHODS OF USE Amgen, Inc (US) 2008-06-11 EP disclosed
WO-2007022380-A2 BIS-ARYL AMIDE COMPOUNDS AND METHODS OF USE AMGEN INC. (US) 2007-02-22 WO disclosed