SCHEMBL4767237

SCHEMBL4767237

Cc1noc(N(COCC[Si](C)(C)C)S(=O)(=O)c2ccccc2-c2ccc(COS(C)(=O)=O)cc2)c1C

nearest known ligand 0.41

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 6/20 0.39
EDNRA P25101 6/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4772907 0.88 EDNRA (0.35) EDNRA
SCHEMBL4774085 0.88 EDNRA (0.36) EDNRA
SCHEMBL5531220 0.88 EDNRA (0.37) EDNRA
SCHEMBL5791432 0.86 EDNRA (0.36) EDNRBEDNRA
SCHEMBL5531005 0.86 EDNRA (0.41) EDNRBEDNRA
SCHEMBL4771374 0.86 EDNRA (0.32) EDNRA
SCHEMBL4770730 0.85 EDNRA (0.38) EDNRA
SCHEMBL4769236 0.85 EDNRA (0.38) EDNRBEDNRA
SCHEMBL4774149 0.84 EDNRA (0.34) EDNRBEDNRA
SCHEMBL4765078 0.84 EDNRA (0.38) EDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2002837-A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-17 EP disclosed
EP-1094816-B1 BIPHENYL SULFONAMIDES AS DUAL ANGIOTENSIN ENDOTHELIN RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2008-12-10 EP disclosed
EP-1741713-A2 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists Bristol-Myers Squibb Company (US) 2007-01-10 EP disclosed
EP-1237888-B1 BIPHENYL SULFONAMIDES AS DUAL ANGIOTENSIN ENDOTHELIN RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2006-09-13 EP disclosed
US-6852745-B2 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists BRISTOL-MYERS SQUIBB COMPANY (US) 2005-02-08 US disclosed
US-6835741-B2 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists BRISTOL-MYERS SQUIBB COMPANY 2004-12-28 US disclosed
US-6638937-B2 As antihypertensive agents; for therapy of disorders related to renal, glomerular and mesangial cell function; therapy of endotoxemia or endotoxin shock as well as hemorrhagic shock; useful in alleviation of pain associated cancer BRISTOL-MYERS SQUIBB CO. 2003-10-28 US disclosed