SCHEMBL4767496

SCHEMBL4767496

CC(C)(C)OC(=O)N1CC(=O)C(=CN)C1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NR1H2 P55055 4/20 0.39
HDAC1 Q13547 1/20 0.38
ESR2 Q92731 1/20 0.37
ADORA1 P30542 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
MAPK1 P28482 1/20 0.36
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
HPGD P15428 1/20 0.35
GPR119 Q8TDV5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15248097 0.85 USP2 (0.41) USP2SMN1; SMN2NR1H2HDAC1ESR2
SCHEMBL20392811 0.83 USP2 (0.39) USP2SMN1; SMN2NR1H2HDAC1ESR2
SCHEMBL31080015 0.82 USP2 (0.50) USP2SMN1; SMN2NR1H2HDAC1ESR2
SCHEMBL1528547 0.81 USP2 (0.38) USP2SMN1; SMN2NR1H2HDAC1ESR2
SCHEMBL1528546 0.81 USP2 (0.38) USP2SMN1; SMN2NR1H2HDAC1ESR2
SCHEMBL827122 0.81 USP2 (0.38) USP2SMN1; SMN2NR1H2HDAC1ESR2
SCHEMBL21588714 0.80 USP2 (0.44) USP2SMN1; SMN2NR1H2HDAC1ESR2
SCHEMBL4768968 0.79 MAPK10 (0.39) USP2SMN1; SMN2NR1H2HDAC1ESR2
SCHEMBL17081081 0.77 USP2 (0.42) USP2SMN1; SMN2NR1H2HDAC1ESR2
SCHEMBL25845889 0.76 NR1H2 (0.47) USP2SMN1; SMN2NR1H2ESR2ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1412078-B1 PROCESSES FOR THE PRODUCTION OF AMINO-PROTECTED DERIVATIVES OF 4-AMINOMETHYLENE-PYRROLIDIN-3-ONE, GEMIFLOXACIN OR A SALT THEREOF LG LIFE SCIENCES LTD (KR) 2008-10-08 EP disclosed
US-7199242-B2 Processes for the production of amino-protected derivatives of 4-aminomethylene-pyrrolidin-3-one and/or 4-aminomethylene-pyrrolidin-3-alkoxyimino derivatives and/or gemifloxacin or a salt thereof LG LIFE SCIENCES LIMITED (KR) 2007-04-03 US disclosed
US-7199242-B2 Processes for the production of amino-protected derivatives of 4-aminomethylene-pyrrolidin-3-one and/or 4-aminomethylene-pyrrolidin-3-alkoxyimino derivatives and/or gemifloxacin or a salt thereof LG LIFE SCIENCES LIMITED (KR) 2007-04-03 US disclosed
US-7199242-B2 Processes for the production of amino-protected derivatives of 4-aminomethylene-pyrrolidin-3-one and/or 4-aminomethylene-pyrrolidin-3-alkoxyimino derivatives and/or gemifloxacin or a salt thereof LG LIFE SCIENCES LIMITED (KR) 2007-04-03 US disclosed
EP-1068182-B1 PROCESS FOR PREPARING A PROTECTED 4-AMINOMETHYL-PYRROLIDIN-3-ONE LG LIFE SCIENCES LTD (KR) 2005-06-08 EP disclosed
US-20050043546-A1 Processes for the production of amino-protected derivatives of 4-aminomethylene-pyrrolidin-3-one and/or 4-aminomethylene-pyrrolidin-3-alkoxyimino derivatives and/or gemifloxacin or a salt thereof LG CHEM, LTD. (KR) 2005-02-24 US disclosed
EP-1412078-A1 PROCESSES FOR THE PRODUCTION OF AMINO-PROTECTED DERIVATIVES OF 4-AMINOMETHYLENE-PYRROLIDIN-3-ONE AND/OR 4-AMINOMETHYLENE-PYRROLIDIN-3-ALKOXYIMINO DERIVATIVES AND/OR GEMIFLOXACIN OR A SALT THEREOF SB Pharmco Puerto Rico Inc (US) 2004-04-28 EP disclosed
WO-2003011450-A1 PROCESSES FOR THE PRODUCTION OF AMINO-PROTECTED DERIVATIVES OF 4-AMINOMETHYLENE-PYRROLIDIN-3-ONE AND/OR 4-AMINOMETHYLENE-PYRROLIDIN-3-ALKOXYIMINO DERIVATIVES AND/OR GEMIFLOXACIN OR A SALT THEREOF LG LIFE SCIENCES LIMITED (KR) 2003-02-13 WO disclosed
US-6307059-B1 PREPARATION OF QUINOLONE ANTIBIOTICS. LG CHEMICAL, LTD (KR) 2001-10-23 US disclosed
WO-2001040163-A1 A PROCESS FOR PRODUCING AMINE COMPOUND WITH t-BUTOXYCARBONYL GROUP KOREA FINE CHEMICAL CO.,LTD. (KR) 2001-06-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050043546-A1 Processes for the production of amino-protected derivatives of 4-aminomethylene-pyrrolidin-3-one and/or 4-aminomethylene-pyrrolidin-3-alkoxyimino derivatives and/or gemifloxacin or a salt thereof CYP4X1, PM20D2, BRIX1 USP2 3909/4885SMN1; SMN2 3131/4885NR1H2 4584/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.