SCHEMBL4769690

SCHEMBL4769690

CCCn1c(=O)c([N+](=O)[O-])c(C=Cc2cnn(Cc3ccccc3C(F)(F)F)c2)n(CC)c1=O

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 18/20 0.52
ADORA1 P30542 14/20 0.52
ADORA2A P29274 11/20 0.52
ADORA3 P0DMS8 5/20 0.40
PLK4 O00444 1/20 0.37
CDK2 P24941 1/20 0.37
IRAK1 P51617 1/20 0.37
RPS6KA3 P51812 1/20 0.37
PLK3 Q9H4B4 1/20 0.37
CSNK1G3 Q9Y6M4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769673 1.00 ADORA2B (0.52) ADORA2BADORA1ADORA2AADORA3PLK4
SCHEMBL4767719 0.95 ADORA2B (0.45) ADORA2BADORA1ADORA2AADORA3
SCHEMBL4767733 0.95 ADORA2B (0.45) ADORA2BADORA1ADORA2AADORA3
SCHEMBL4770754 0.92 ADORA2B (0.48) ADORA2BADORA1ADORA2AADORA3
SCHEMBL4770747 0.92 ADORA2B (0.48) ADORA2BADORA1ADORA2AADORA3
SCHEMBL4766139 0.91 ADORA2B (0.49) ADORA2BADORA1ADORA2AADORA3
SCHEMBL4769328 0.90 ADORA2B (0.49) ADORA2BADORA1ADORA2AADORA3
SCHEMBL4769321 0.90 ADORA2B (0.49) ADORA2BADORA1ADORA2AADORA3
SCHEMBL4763384 0.88 ADORA2B (0.44) ADORA2BADORA1ADORA2AADORA3
SCHEMBL4766145 0.88 ADORA2B (0.41) ADORA2BADORA1ADORA2AADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed