SCHEMBL4769852

SCHEMBL4769852

COc1ccc(NC2CCCN2C(=O)OC(C)(C)C)cc1Cl

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 5/20 0.50
SMN1; SMN2 Q16637 2/20 0.47
GAA P10253 1/20 0.47
ALDH1A1 P00352 4/20 0.46
MAPT P10636 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
NPC1 O15118 1/20 0.46
MAPK1 P28482 1/20 0.46
GPR35 Q9HC97 1/20 0.46
GPR55 Q9Y2T6 1/20 0.46
HPGD P15428 1/20 0.45
EPHA2 P29317 1/20 0.43
KDR P35968 1/20 0.43
EPHB4 P54760 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769848 1.00 MALT1 (0.50) MALT1SMN1; SMN2GAAALDH1A1MAPT
SCHEMBL4764237 0.89 ALDH1A1 (0.49) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL4764235 0.89 ALDH1A1 (0.49) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL330988 0.86 ALDH1A1 (0.49) MALT1GAAALDH1A1MAPTMEN1
SCHEMBL330987 0.86 ALDH1A1 (0.49) MALT1GAAALDH1A1MAPTMEN1
SCHEMBL30968029 0.83 MEN1 (0.46) SMN1; SMN2ALDH1A1MAPTMEN1KMT2A
SCHEMBL4790229 0.82 ALDH1A1 (0.65) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL4790228 0.82 ALDH1A1 (0.65) ALDH1A1MAPTMEN1KMT2ANPC1
SCHEMBL329897 0.80 ALDH1A1 (0.59) MALT1SMN1; SMN2GAAALDH1A1MAPT
SCHEMBL329898 0.80 ALDH1A1 (0.59) MALT1SMN1; SMN2GAAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881975-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-01-30 EP disclosed
WO-2006121218-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-11-16 WO disclosed