SCHEMBL4771317

SCHEMBL4771317

CC(=O)N1CCC(C(=O)N(CCCN2CCC(N(C)S(=O)(=O)c3ccc(F)cc3)CC2)c2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.79

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.79
KCNH2 Q12809 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4768540 0.91 CCR5 (0.75) CCR5KCNH2
SCHEMBL4768594 0.88 CCR5 (1.00) CCR5KCNH2
SCHEMBL4773958 0.87 CCR5 (0.81) CCR5KCNH2
SCHEMBL4777027 0.86 CCR5 (0.83) CCR5KCNH2
SCHEMBL4775650 0.84 CCR5 (0.80) CCR5KCNH2
SCHEMBL4775171 0.84 CCR5 (1.00) CCR5KCNH2
SCHEMBL4775616 0.83 CCR5 (0.78) CCR5KCNH2
Hydrochloric Acid SCHEMBL4771685 0.83 CCR5 (0.98) CCR5KCNH2
SCHEMBL4768104 0.83 CCR5 (0.74) CCR5KCNH2
SCHEMBL4777222 0.82 CCR5 (1.00) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7348324-B2 Cyclic amine compounds as CCR5 antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-03-25 US disclosed
EP-1886994-A1 Cyclic amine compounds as CCR5 antagonists Takeda Pharmaceutical Company Limited (JP) 2008-02-13 EP disclosed
US-6562978-B1 N-(3-(4-(4-(Aminocarbonyl)benzyl)-1-piperidinyl)propyl)-N-(3, 4-dichlorophenyl)-1-(methylsulfonyl)-4-piperidinecarboxamide or a salt thereof for treatment of AIDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-13 US disclosed