SCHEMBL4771530

SCHEMBL4771530

CCOC(=O)c1cn(-c2ccc3c(c2)CCC3)c2nc(N(c3ccccc3)N3CCNCC3)ncc2c1=O

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 20/20 0.57
NTRK1 P04629 2/20 0.43
KIT P10721 2/20 0.43
SRC P12931 2/20 0.43
FLT3 P36888 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771164 0.88 CSF1R (0.63) CSF1RNTRK1KITSRCFLT3
SCHEMBL4572926 0.84 CSF1R (0.53) CSF1RNTRK1KITSRCFLT3
SCHEMBL4775794 0.79 CSF1R (0.55) CSF1RNTRK1KITSRCFLT3
SCHEMBL3530794 0.79 CSF1R (0.86) CSF1RNTRK1KITSRCFLT3
SCHEMBL4775457 0.79 CSF1R (0.57) CSF1RNTRK1KITSRCFLT3
SCHEMBL3525502 0.78 CSF1R (0.75) CSF1RNTRK1KITSRCFLT3
SCHEMBL3529843 0.78 CSF1R (0.58) CSF1RNTRK1KITSRCFLT3
SCHEMBL3289970 0.78 CSF1R (0.65) CSF1RNTRK1KITSRCFLT3
SCHEMBL3289501 0.77 CSF1R (0.65) CSF1RNTRK1KITSRCFLT3
SCHEMBL3533106 0.77 CSF1R (0.65) CSF1RNTRK1KITSRCFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937681-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-07-02 EP disclosed
WO-2007033232-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-22 WO disclosed