SCHEMBL4771748

SCHEMBL4771748

COc1ccc(-c2cc(-c3ccc(OC)cc3Cl)cn2-c2ccc(OC)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MARS1 P56192 1/20 0.46
RAD51 Q06609 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
MEN1 O00255 1/20 0.40
TP53 P04637 1/20 0.40
HPGD P15428 1/20 0.40
ALOX12 P18054 1/20 0.40
KMT2A Q03164 1/20 0.40
RPA1 P27694 1/20 0.40
FASN P49327 1/20 0.40
PTGS1 P23219 3/20 0.40
PTGS2 P35354 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
THPO P40225 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780371 0.80 HSP90AA1 (0.39) MARS1MEN1KMT2AFASNCYP1A2
SCHEMBL4771806 0.78 ESRRA (0.40) MARS1RAD51MAPTRAB9ARXFP1
SCHEMBL4778866 0.75 CHRNA7 (0.42) MARS1MEN1TP53HPGDKMT2A
SCHEMBL4778476 0.72 TP53 (0.43) MARS1MEN1TP53HPGDKMT2A
SCHEMBL12325069 0.72 HSP90AA1 (0.56) MAPTRAB9AMEN1HPGDKMT2A
SCHEMBL4779727 0.70 TP53 (0.41) MARS1MAPTRAB9AMEN1TP53
SCHEMBL28303202 0.70 ESR2 (0.57) MAPTRAB9AMEN1TP53ALOX12
SCHEMBL9732916 0.70 CYP2A6 (0.50) MAPTRAB9AMEN1TP53HPGD
SCHEMBL4779710 0.70 TP53 (0.39) MARS1MEN1TP53HPGDKMT2A
SCHEMBL31265226 0.67 GSK3B (0.48) MAPTRAB9AMEN1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1889617-A1 Triphenyl modified 5-membered heterocycles and their use as anticancer and antiflammatory agents Freie Universität Berlin (DE) 2008-02-20 EP claimed
EP-1889617-A1 Triphenyl modified 5-membered heterocycles and their use as anticancer and antiflammatory agents Freie Universität Berlin (DE) 2008-02-20 EP disclosed