SCHEMBL4771806

SCHEMBL4771806

COc1ccc(-c2c(C)c(-c3ccc(OC)cc3Cl)cn2-c2ccc(OC)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRA P11474 2/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
MAPT P10636 2/20 0.40
RAD51 Q06609 1/20 0.40
RAB9A P51151 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
GRIK1 P39086 1/20 0.39
GRIK2 Q13002 1/20 0.39
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
TP53 P04637 1/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
GAA P10253 1/20 0.39
ATM Q13315 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771748 0.78 MARS1 (0.46) ESRRAPTGS1PTGS2MAPTRAD51
SCHEMBL12325069 0.73 HSP90AA1 (0.56) MAPTRAB9AKMT2AMEN1HPGD
SCHEMBL4778866 0.73 CHRNA7 (0.42) PTGS1PTGS2KMT2AMEN1TP53
SCHEMBL4778476 0.68 TP53 (0.43) PTGS1PTGS2KMT2AMEN1TP53
SCHEMBL7906452 0.67 HSP90AA1 (0.50) MAPTRAB9AKMT2AMEN1HPGD
SCHEMBL4779727 0.66 TP53 (0.41) MAPTRAB9AKMT2AMEN1TP53
SCHEMBL5478017 0.66 HSP90AA1 (0.43) MAPTRAB9AKMT2AMEN1HPGD
SCHEMBL28303202 0.65 ESR2 (0.57) MAPTRAB9AKMT2AMEN1TP53
SCHEMBL9732916 0.65 CYP2A6 (0.50) MAPTRAB9AKMT2AMEN1TP53
SCHEMBL14055298 0.65 HSP90AA1 (0.55) MAPTRAB9AKMT2AMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1889617-A1 Triphenyl modified 5-membered heterocycles and their use as anticancer and antiflammatory agents Freie Universität Berlin (DE) 2008-02-20 EP claimed
WO-2008006626-A1 TRIPHENYL MODIFIED 5-MEMBERED HETEROCYCLES AND THEIR USE AS ANTICANCER AND ANTIINFLAMMATORY AGENTS FREIE UNIVERSITÄT BERLIN (DE) 2008-01-17 WO claimed
EP-1889617-A1 Triphenyl modified 5-membered heterocycles and their use as anticancer and antiflammatory agents Freie Universität Berlin (DE) 2008-02-20 EP disclosed