SCHEMBL4771823

SCHEMBL4771823

CCOC(=O)c1cc(-c2ccncc2)[nH]c1CC(NC(=O)OC(C)(C)C)C1CC1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GCGR P47871 2/20 0.46
CDC7 O00311 4/20 0.40
AAK1 Q2M2I8 2/20 0.40
MAPK14 Q16539 1/20 0.37
CDK5 Q00535 5/20 0.37
CDK5R1 Q15078 5/20 0.37
MMP2 P08253 1/20 0.37
MMP13 P45452 1/20 0.37
MMP14 P50281 1/20 0.37
CASP1 P29466 1/20 0.36
BUB1 O43683 1/20 0.35
ACACB O00763 1/20 0.35
ACACA Q13085 1/20 0.35
GSK3B P49841 1/20 0.35
ABCB1 P08183 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4830885 0.96 GCGR (0.44) GCGRCDC7AAK1MAPK14CDK5
SCHEMBL4767710 0.86 GCGR (0.49) GCGRCDC7AAK1MAPK14CDK5
SCHEMBL6466255 0.85 KDM4E (0.35) MMP13CASP1ACACBACACA
SCHEMBL4774859 0.85 GCGR (0.48) GCGRCDC7AAK1MAPK14CDK5
SCHEMBL4767661 0.82 GCGR (0.46) GCGRCDC7AAK1MAPK14CDK5
SCHEMBL4771352 0.82 ATM (0.46) GCGRCDC7AAK1CDK5CDK5R1
Hydrochloric Acid SCHEMBL4775133 0.80 GCGR (0.52) GCGRCDC7MAPK14CDK5CDK5R1
SCHEMBL4768810 0.79 GCGR (0.51) GCGRCDC7AAK1MAPK14CDK5
Hydrochloric Acid SCHEMBL4765927 0.75 GCGR (0.49) GCGRCDC7MAPK14CDK5CDK5R1
SCHEMBL5346356 0.75 GCGR (0.53) GCGRCDC7AAK1MAPK14CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1660085-B1 PYRIDYLPYRROLE DERIVATIVES ACTIVE AS KINASE INHIBITORS PFIZER ITALIA SRL (IT) 2008-10-15 EP disclosed