SCHEMBL5346356

SCHEMBL5346356

CCOC(=O)c1cc(-c2ccncc2)[nH]c1C(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 3/20 0.53
MAPK14 Q16539 1/20 0.42
CDK5 Q00535 3/20 0.42
CDK5R1 Q15078 3/20 0.42
CASP1 P29466 1/20 0.42
CDC7 O00311 5/20 0.41
MMP2 P08253 1/20 0.40
MMP13 P45452 1/20 0.40
MMP14 P50281 1/20 0.40
PKN1 Q16512 1/20 0.39
PKN2 Q16513 1/20 0.39
AAK1 Q2M2I8 2/20 0.39
ROCK2 O75116 1/20 0.39
PIM1 P11309 1/20 0.39
GSK3B P49841 1/20 0.39
HIPK2 Q9H2X6 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4768810 0.80 GCGR (0.51) GCGRMAPK14CDK5CDK5R1CASP1
SCHEMBL4775802 0.78 GCGR (0.49) GCGRMAPK14CDK5CDK5R1CASP1
SCHEMBL4767710 0.78 GCGR (0.49) GCGRMAPK14CDK5CDK5R1CASP1
SCHEMBL4774859 0.77 GCGR (0.48) GCGRMAPK14CDK5CDK5R1CASP1
SCHEMBL4174038 0.75 GCGR (0.66) GCGRMAPK14CDK5CDK5R1CASP1
SCHEMBL4182065 0.75 GCGR (0.86) GCGRMAPK14CASP1CDC7MMP2
SCHEMBL4771823 0.75 GCGR (0.46) GCGRMAPK14CDK5CDK5R1CASP1
SCHEMBL4767661 0.75 GCGR (0.46) GCGRMAPK14CDK5CDK5R1CDC7
SCHEMBL15230740 0.74 PIM1 (0.54) PIM1
SCHEMBL4771352 0.74 ATM (0.46) GCGRCDK5CDK5R1CDC7AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096334-A1 PYRROLOPYRROLONES ACTIVE AS KINASE INHIBITORS PFIZER ITALIA SRL (IT) 2007-08-30 WO disclosed