SCHEMBL4773463

SCHEMBL4773463

CCCOc1ccc(C(=O)N[C@H](CCO)Cc2ccc(-c3cn(C)c(C(C)=O)n3)cc2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CENPE Q02224 2/20 0.45
GCGR P47871 2/20 0.38
GIPR P48546 2/20 0.38
TAS1R3 Q7RTX0 4/20 0.37
TAS1R1 Q7RTX1 4/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
PPARG P37231 5/20 0.36
NLRP3 Q96P20 1/20 0.36
ITGB1 P05556 1/20 0.35
ITGA4 P13612 1/20 0.35
ITGB7 P26010 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKACA P17612 1/20 0.35
RPS6KB1 P23443 1/20 0.35
IRAK1 P51617 1/20 0.35
PRKX P51817 1/20 0.35
LIMK1 P53667 1/20 0.35
PRKG2 Q13237 1/20 0.35
ROCK1 Q13464 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2630622 0.94 CENPE (0.46) CENPETAS1R3TAS1R1ALDH1A1MAPT
SCHEMBL3233585 0.92 CENPE (0.41) CENPEGCGRGIPRTAS1R3TAS1R1
SCHEMBL3223158 0.91 CENPE (0.39) CENPEGCGRGIPRTAS1R3TAS1R1
SCHEMBL3228196 0.89 CENPE (0.42) CENPEGCGRGIPRTAS1R3TAS1R1
SCHEMBL4435296 0.89 CENPE (0.41) CENPEGCGRGIPRTAS1R3TAS1R1
SCHEMBL2104300 0.89 CENPE (0.55) CENPETAS1R3TAS1R1ITGA4ITGB7
SCHEMBL2104302 0.89 CENPE (0.55) CENPETAS1R3TAS1R1ITGA4ITGB7
SCHEMBL3229991 0.89 CENPE (0.45) CENPEGCGRGIPRTAS1R3TAS1R1
SCHEMBL3229222 0.88 CENPE (0.43) CENPEGCGRGIPRTAS1R3TAS1R1
SCHEMBL3219631 0.88 CENPE (0.43) CENPEGCGRGIPRTAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742907-A4 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS INC (US) 2008-01-02 EP disclosed
EP-1742907-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2007-01-17 EP disclosed
WO-2005107762-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2005-11-17 WO disclosed