SCHEMBL4773992

SCHEMBL4773992

CS(=O)(=O)Nc1cccnc1N1CC2C(C1)C2NC(=O)Nc1cccc2cnccc12

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 15/20 0.45
ROCK2 O75116 4/20 0.44
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
CDK5 Q00535 1/20 0.43
CYP3A4 P08684 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776171 0.88 TRPV1 (0.47) TRPV1ROCK2CCNE1CDK2CDK5
SCHEMBL4778071 0.85 CCNE1 (0.46) TRPV1CCNE1CDK2CDK5CYP3A4
SCHEMBL4777964 0.84 TRPV1 (0.47) TRPV1CCNE1CDK2CDK5CYP3A4
SCHEMBL4776314 0.79 TRPV1 (0.56) TRPV1
SCHEMBL4781057 0.77 TRPV1 (0.55) TRPV1CYP3A4
SCHEMBL4773951 0.76 TRPV1 (0.56) TRPV1CYP3A4
SCHEMBL4773955 0.76 TRPV1 (0.59) TRPV1
SCHEMBL4779491 0.76 TRPV1 (0.51) TRPV1CCNE1CDK2CDK5
SCHEMBL4780302 0.76 TRPV1 (0.52) TRPV1CYP3A4
SCHEMBL4779427 0.75 EPHX2 (0.51) TRPV1CCNE1CDK2CDK5CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008010061-A2 3-AZABICYCLO [3.1.0] HEXANE VANILLOID RECEPTOR LIGANDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESSES FOR THEIR PREPARATION GLENMARK PHARMACEUTICALS S.A. (US) 2008-01-24 WO claimed
WO-2008010061-A2 3-AZABICYCLO [3.1.0] HEXANE VANILLOID RECEPTOR LIGANDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESSES FOR THEIR PREPARATION GLENMARK PHARMACEUTICALS S.A. (US) 2008-01-24 WO disclosed