SCHEMBL4774059

SCHEMBL4774059

CN(C)Cc1ccc(-c2cc3c(N(Cc4ccccc4)C4=COCO4)ncnc3[nH]2)cc1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 17/20 0.58
EGFR P00533 14/20 0.57
PRMT5 O14744 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4764400 0.91 CSF1R (0.53) CSF1REGFR
SCHEMBL4766640 0.91 CSF1R (0.65) CSF1REGFR
SCHEMBL4766600 0.87 KDR (0.56) CSF1REGFRPRMT5
SCHEMBL4764640 0.86 KDR (0.49) CSF1REGFRPRMT5
SCHEMBL4763953 0.85 CSF1R (0.57) CSF1REGFRPRMT5
SCHEMBL4808322 0.72 PRMT5 (0.57) CSF1REGFRPRMT5
SCHEMBL4767171 0.69 EGFR (0.77) CSF1REGFR
SCHEMBL27585232 0.69 EGFR (0.77) CSF1REGFR
SCHEMBL30921904 0.69 EGFR (1.00) CSF1REGFR
SCHEMBL4766838 0.68 CSF1R (0.60) CSF1REGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1416935-B1 4-AMINO-6-PHENYL-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES NOVARTIS AG (CH) 2008-03-12 EP claimed
US-7244729-B2 4-amino-6-phenyl-pyrrolo[2,3-d]pyrimidine derivatives NOVARTIS AG (CH) 2007-07-17 US claimed
US-20040248911-A1 7H-pyrrolo[2,3-d]pyrimidine derivatives BOLD GUIDO (CH) 2004-12-09 US claimed
US-20040242600-A1 4-amino-6-phenyl-pyrrolo[2,3-d]pyrimidine derivatives NOVARTIS AG (CH) 2004-12-02 US claimed
EP-1416935-B1 4-AMINO-6-PHENYL-PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES NOVARTIS AG (CH) 2008-03-12 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040248911-A1 7H-pyrrolo[2,3-d]pyrimidine derivatives DPYD, DHPS, TYMP CSF1R 3024/4885EGFR 3391/4885PRMT5 684/4885
US-20040242600-A1 4-amino-6-phenyl-pyrrolo[2,3-d]pyrimidine derivatives DPYD, TYMP, TYMS CSF1R 3516/4885EGFR 2694/4885PRMT5 345/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.