SCHEMBL4774460

SCHEMBL4774460

CCc1c(Cl)nc(C2CCCCC2)nc1NCc1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 11/20 0.65
PDE5A O76074 2/20 0.61
PDE4A P27815 3/20 0.51
PDE4B Q07343 3/20 0.51
PDE4C Q08493 3/20 0.51
PDE4D Q08499 3/20 0.51
CHRM3 P20309 1/20 0.51
F2 P00734 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4095293 0.76 PDE5A (1.00) PDE10APDE5APDE4APDE4BPDE4C
SCHEMBL4776578 0.76 PDE10A (0.48) PDE10APDE4APDE4BPDE4CPDE4D
SCHEMBL7422996 0.74 PDE5A (0.61) PDE10APDE5APDE4APDE4BPDE4C
SCHEMBL7425485 0.74 PDE5A (0.64) PDE10APDE5APDE4APDE4BPDE4C
SCHEMBL4794212 0.73 PDE5A (0.46) PDE10APDE5APDE4APDE4BPDE4C
Bicarbonate SCHEMBL7016629 0.71 PDE5A (0.57) PDE10APDE5APDE4APDE4BPDE4C
Bicarbonate SCHEMBL7017171 0.71 PDE10A (0.52) PDE10APDE5APDE4APDE4BPDE4C
SCHEMBL11104154 0.71 EGFR (0.53) PDE5APDE4APDE4BPDE4CPDE4D
Bicarbonate SCHEMBL7017039 0.70 PDE5A (0.59) PDE10APDE5APDE4APDE4BPDE4C
SCHEMBL1609704 0.70 PDE10A (0.62) PDE10APDE5APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed