SCHEMBL4776578

SCHEMBL4776578

CCc1c(Cl)nc(C2CCCCC2)nc1Cl

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 13/20 0.48
CHRM3 P20309 5/20 0.35
PDE4A P27815 3/20 0.35
PDE4B Q07343 3/20 0.35
PDE4C Q08493 3/20 0.35
PDE4D Q08499 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NR1I2 O75469 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4429704 0.90 PDE10A (0.59) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL4774460 0.76 PDE10A (0.65) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL4421489 0.75 PDE10A (0.83) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL909354 0.73 PDE10A (0.64) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL4420885 0.73 PDE10A (0.57) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL6919137 0.72 PDE10A (0.40) PDE10A
SCHEMBL4419024 0.71 PDE10A (0.83) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL6396181 0.71 CHRM3 (0.43) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL27846371 0.70 PDE10A (0.83) PDE10ACHRM3PDE4APDE4BPDE4C
SCHEMBL18520713 0.70 PDE10A (0.43) PDE10ACHRM3PDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed