SCHEMBL4774462

SCHEMBL4774462

Cc1c(C(=O)Nc2ccc3c(c2)CCN(C2CCC2)CC3)cnn1-c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 15/20 0.59
NPC1 O15118 14/20 0.59
PKM P14618 3/20 0.59
HPGD P15428 1/20 0.53
NFKB1 P19838 1/20 0.53
NFKB2 Q00653 1/20 0.53
RELA Q04206 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
POLB P06746 1/20 0.53
NAMPT P43490 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
TRPV4 Q9HBA0 1/20 0.49
PARP1 P09874 1/20 0.47
ROCK1 Q13464 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4771045 0.92 RAB9A (0.53) RAB9ANPC1PKMHPGDNFKB1
SCHEMBL4768108 0.91 NPC1 (0.51) RAB9ANPC1PKMHPGDNFKB1
SCHEMBL4765305 0.91 RAB9A (0.48) RAB9ANPC1PKMHPGDNFKB1
Hydrochloric Acid SCHEMBL4774495 0.90 RAB9A (0.47) RAB9ANPC1PKMHPGDNFKB1
Hydrochloric Acid SCHEMBL4776625 0.90 NPC1 (0.50) RAB9ANPC1PKMHPGDNFKB1
SCHEMBL4772163 0.89 NPC1 (0.57) RAB9ANPC1PKMPOLBKMT2A
SCHEMBL4768367 0.89 NPC1 (0.48) RAB9ANPC1PKMHPGDNFKB1
Hydrochloric Acid SCHEMBL4770710 0.88 NPC1 (0.47) RAB9ANPC1PKMHPGDNFKB1
SCHEMBL4765359 0.88 NPC1 (0.44) RAB9ANPC1PKMNFKB1NFKB2
Hydrochloric Acid SCHEMBL4772031 0.87 NPC1 (0.43) RAB9ANPC1PKMNFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713778-B1 BENZAZEPINE DERIVATIVES AS HISTAMINE H3 ANTAGONISTS GLAXO GROUP LTD (GB) 2008-01-16 EP claimed