SCHEMBL477477

SCHEMBL477477

OC(c1ccccc1)c1ccc(F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
KMT2A Q03164 1/20 0.47
ATM Q13315 1/20 0.47
LMNA P02545 2/20 0.46
HPGD P15428 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HTT P42858 2/20 0.46
USP2 O75604 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
NPC1 O15118 1/20 0.43
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21542545 1.00 EPHX1 (0.48) EPHX1SMN1; SMN2KMT2AATMLMNA
SCHEMBL21542539 1.00 EPHX1 (0.48) EPHX1SMN1; SMN2KMT2AATMLMNA
SCHEMBL4532015 0.93 CA1 (0.55) EPHX1SMN1; SMN2KMT2AATMLMNA
SCHEMBL597442 0.89 IDO1 (0.46) SMN1; SMN2KMT2AATMLMNAALDH1A1
SCHEMBL11640483 0.89 KMT2A (0.51) EPHX1KMT2AATMALDH1A1CA12
SCHEMBL8671295 0.87 SMN1; SMN2 (0.58) SMN1; SMN2LMNACA12CA1CA2
SCHEMBL11602058 0.85 CYP19A1 (0.49) EPHX1SMN1; SMN2KMT2ALMNAHPGD
Diphenylmethanol SCHEMBL10868602 0.84 SMN1; SMN2 (0.61) SMN1; SMN2LMNACA12CA1CA2
Diphenylmethanol SCHEMBL41571 0.84 SMN1; SMN2 (0.61) SMN1; SMN2LMNACA12CA1CA2
Diphenylmethanol SCHEMBL6434457 0.84 SMN1; SMN2 (0.61) SMN1; SMN2LMNACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 90 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117362236-B Synthesis method of flumazenil 江苏远恒药业有限公司 2024-05-03 CN claimed
CN-117362236-A Synthesis method of flumazenil 江苏远恒药业有限公司 2024-01-09 CN claimed
CN-112517060-B Catalyst, application and synthesis method of 4-hydroxycoumarin derivative 山东农业大学 2022-03-25 CN claimed
EP-2665703-B1 ENANTIOMER (R) OF LAUFLUMIDE IN MEHR ALS 95%ee NLS PHARMA AG (CH) 2017-12-06 EP claimed
EP-2665703-A1 LAUFLUMIDE AND THE ENANTIOMERS THEREOF, METHOD FOR PREPARING SAME AND THERAPEUTIC USES THEREOF Assistance Publique Hôpitaux De Paris (FR) 2013-11-27 EP claimed
US-20130295196-A1 LAUFLUMIDE AND THE ENANTIOMERS THEREOF, METHOD FOR PREPARING SAME AND THERAPEUTIC USES THEREOF ASSISTANCE PUBLIQUE-HOPITAUX DE PARIS (FR) 2013-11-07 US claimed
WO-2012098235-A1 LAUFLUMIDE AND THE ENANTIOMERS THEREOF, METHOD FOR PREPARING SAME AND THERAPEUTIC USES THEREOF ASSISTANCE PUBLIQUE - HOPITAUX DE PARIS (FR) 2012-07-26 WO claimed
EP-0686635-A1 Pyridylthiazolidinecarboxylic acid amide derivatives, their preparation and their therapeutic uses Sankyo Company Limited (JP) 1995-12-13 EP claimed
US-5470851-A Antihistamine, anticoagulants SANKYO COMPANY, LIMITED (JP) 1995-11-28 US claimed
EP-0549364-A1 Pyridylthiazolidinecarboxylic acid amide derivatives, their preparation and their therapeutic uses Sankyo Company Limited (JP) 1993-06-30 EP claimed
EP-4583876-A1 COMBINATION OF A T CELL THERAPY AND CONTINUOUS OR INTERMITTENT DGK INHIBITOR DOSING Juno Therapeutics, Inc. (US) 2025-07-16 EP disclosed
CN-120152717-A Combination of T cell therapy and continuous or intermittent DGK inhibitor administration 朱诺治疗学股份有限公司 2025-06-13 CN disclosed
CN-112654621-B Substituted naphthyridinone compounds useful as T cell activators 百时美施贵宝公司 2024-05-14 CN disclosed
CN-117362236-B Synthesis method of flumazenil 江苏远恒药业有限公司 2024-05-03 CN disclosed
CN-117362236-B Synthesis method of flumazenil 江苏远恒药业有限公司 2024-05-03 CN disclosed
US-4916058-A CHROMOGENS KYOWA MEDEX CO., LTD. (JP) 1990-04-10 US disclosed
US-4874765-A 1,4-Disubstituted piperazines having dopaminergic activity RICHTER GEDEON VEGYESZETI GYAR (HU) 1989-10-17 US disclosed
EP-0243903-A1 Optionally substituted 1-(omega[bis(phenyl)-alcoxy]-alkyl)-4-(alkenyl)piperazines and -4-(alkynyl)piperazines, process for their preparation and medicines containing them Richter Gedeon Vegyészeti Gyár R.T. (HU) 1987-11-04 EP disclosed
EP-0124287-A2 Method and test composition for determination of hydrogen peroxide Kyowa Medex Co. Ltd. (JP) 1984-11-07 EP disclosed
US-4202896-A DOPAMINERGIC ACTIVITY GIST-BROCADES N.V. (NL) 1980-05-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130295196-A1 LAUFLUMIDE AND THE ENANTIOMERS THEREOF, METHOD FOR PREPARING SAME AND THERAPEUTIC USES THEREOF HCRTR2, HNMT, CYP2U1 EPHX1 530/4885SMN1; SMN2 656/4885KMT2A 110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.