SCHEMBL4774906

SCHEMBL4774906

O=C(c1ccccn1)c1ncc(Cl)cc1NS(=O)(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53
ALDH1A1 P00352 1/20 0.53
SLC40A1 Q9NP59 1/20 0.51
CLK1 P49759 1/20 0.50
GAA P10253 1/20 0.50
CCR2 P41597 3/20 0.49
CCR1 P32246 2/20 0.49
CCR4 P51679 2/20 0.49
TLR7 Q9NYK1 1/20 0.48
CKS1B P61024 2/20 0.47
SKP2 Q13309 2/20 0.47
CYP2C9 P11712 1/20 0.47
ACLY P53396 1/20 0.46
TSHR P16473 1/20 0.46
KDM1A O60341 2/20 0.45
CCR9 P51686 1/20 0.44
SLC20A2 Q08357 1/20 0.43
SLC20A1 Q8WUM9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29888331 0.86 CYP2C9 (0.63) KMT2AMEN1ALDH1A1CCR2CYP2C9
SCHEMBL306095 0.86 CYP2C9 (0.63) KMT2AMEN1ALDH1A1CCR2CYP2C9
SCHEMBL10223198 0.82 CCR2 (0.47) KMT2AMEN1SLC40A1CLK1GAA
SCHEMBL10223220 0.82 MEN1 (0.53) KMT2AMEN1SLC40A1CLK1GAA
SCHEMBL10223329 0.81 MEN1 (0.52) KMT2AMEN1SLC40A1GAACCR2
SCHEMBL12594346 0.80 MEN1 (0.52) KMT2AMEN1CCR2CCR4CYP2C9
SCHEMBL1762318 0.79 CYP2C9 (0.58) KMT2AMEN1SLC40A1CLK1GAA
SCHEMBL4799079 0.79 CCR2 (0.46) KMT2AMEN1SLC40A1CLK1GAA
SCHEMBL305413 0.78 CCR2 (0.53) KMT2AMEN1SLC40A1CLK1GAA
SCHEMBL4778194 0.78 CYP2C9 (0.44) KMT2AMEN1SLC40A1CLK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008008431-A2 HETEROARYL SULFONAMIDES AND CCR2/CCR9 CHEMOCENTRYX, INC. (US) 2008-01-17 WO disclosed