SCHEMBL4774956

SCHEMBL4774956

C[C@H](Nc1ccc(Cl)cc1Cl)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.54
CA14 Q9ULX7 1/20 0.54
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
KDM4E B2RXH2 3/20 0.44
PDK1 Q15118 1/20 0.44
PDK2 Q15119 1/20 0.44
PDK3 Q15120 1/20 0.44
PDK4 Q16654 1/20 0.44
USP2 O75604 1/20 0.44
HPGD P15428 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
KDM4C Q9H3R0 1/20 0.44
ALDH1A1 P00352 4/20 0.44
NPC1 O15118 2/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4774951 1.00 CA1 (0.54) CA1CA14TAS1R3TAS1R1KDM4E
SCHEMBL11201439 0.83 CA1 (0.51) CA1CA14TAS1R3TAS1R1KDM4E
SCHEMBL11201438 0.83 CA1 (0.51) CA1CA14TAS1R3TAS1R1KDM4E
SCHEMBL20798060 0.83 KDM4C (0.42) CA1CA14KDM4EKDM4CALDH1A1
SCHEMBL20798059 0.83 KDM4C (0.42) CA1CA14KDM4EKDM4CALDH1A1
SCHEMBL24613827 0.80 CA1 (0.51) CA1CA14TAS1R3TAS1R1KDM4E
SCHEMBL7298206 0.80 PDE2A (0.49) CA1KDM4ENPSR1ALDH1A1LMNA
SCHEMBL7298210 0.80 PDE2A (0.49) CA1KDM4ENPSR1ALDH1A1LMNA
SCHEMBL5022885 0.79 CXCL8 (0.50) TAS1R3TAS1R1KDM4EHPGDNPSR1
SCHEMBL2941689 0.79 CXCL8 (0.50) TAS1R3TAS1R1KDM4EHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3374520-A1 BIOSENSORS Yissum Research and Development Company of the Hebrew University of Jerusalem Ltd. (IL) 2018-09-19 EP claimed
WO-2017081684-A1 BIOSENSORS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD (IL) 2017-05-18 WO claimed
EP-1996550-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES Novartis AG (CH) 2008-12-03 EP disclosed
WO-2007038459-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES NOVARTIS AG (CH) 2007-04-05 WO disclosed