SCHEMBL4774972

SCHEMBL4774972

Nc1nc(N2CCOCC2)c2nc(-c3c(Cl)cccc3Cl)cnc2n1.Nc1nc(N2CCOCC2)c2nc(-c3ccc(C(F)(F)F)cc3C(F)(F)F)cnc2n1.Nc1nc(N2CCOCC2)c2nc(-c3ccc(F)cc3Cl)cnc2n1.Nc1nc(N2CCOCC2)c2nc(-c3ccc(F)cc3F)cnc2n1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.45
ALOX5AP P20292 6/20 0.36
FEN1 P39748 6/20 0.36
LRRK2 Q5S007 1/20 0.35
BRAF P15056 3/20 0.35
RAF1 P04049 2/20 0.35
PIK3CA P42336 3/20 0.34
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
PIK3R1 P27986 1/20 0.33
PTPN1 P18031 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781242 0.89 NOS1 (0.56) NOS1ALOX5APFEN1LRRK2PIK3CA
SCHEMBL3757090 0.84 NOS1 (0.59) NOS1ALOX5APFEN1PIK3CAPIK3R1
SCHEMBL3766398 0.83 NOS1 (0.58) NOS1ALOX5APFEN1BRAFPIK3CA
SCHEMBL3764131 0.82 NOS1 (0.61) NOS1LRRK2PIK3CA
SCHEMBL4781574 0.81 NOS1 (0.56) NOS1PIK3CACNR1CNR2
SCHEMBL3758139 0.81 NOS1 (0.63) NOS1ALOX5APFEN1LRRK2PIK3CA
SCHEMBL3763980 0.78 NOS1 (0.70) NOS1PIK3CACNR2
SCHEMBL3760937 0.75 NOS1 (0.68) NOS1PIK3CACNR2PIK3R1PTPN1
SCHEMBL3760198 0.74 NOS1 (0.63) NOS1LRRK2PIK3CA
SCHEMBL3759317 0.74 NOS1 (0.72) NOS1LRRK2PIK3CACNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009079-A2 SUBSTITUTED PTERIDINES USEFUL FOR THE TREATMENT AND PREVENTION OF VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed