SCHEMBL4774986

SCHEMBL4774986

CCn1cc(-c2ccc(CC(O)CCNC(=O)c3ccc(OC(C)C)c(C#N)c3)cc2)nc1CC(C)O

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CENPE Q02224 2/20 0.50
S1PR1 P21453 7/20 0.41
NPC1 O15118 1/20 0.37
S1PR5 Q9H228 2/20 0.37
S1PR3 Q99500 1/20 0.37
XDH P47989 2/20 0.37
MAPT P10636 2/20 0.36
TP53 P04637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13584373 0.83 CENPE (0.52) CENPES1PR1S1PR5S1PR3XDH
SCHEMBL4767596 0.81 CENPE (0.44) CENPES1PR1NPC1S1PR5S1PR3
SCHEMBL13584416 0.80 CENPE (0.62) CENPES1PR1S1PR5S1PR3XDH
SCHEMBL4837737 0.80 CENPE (0.49) CENPES1PR1S1PR5S1PR3XDH
SCHEMBL3461278 0.78 CENPE (0.66) CENPES1PR1S1PR5S1PR3XDH
SCHEMBL4838728 0.77 CENPE (0.45) CENPES1PR1S1PR5S1PR3XDH
SCHEMBL3461702 0.76 CENPE (0.69) CENPES1PR1S1PR5S1PR3XDH
SCHEMBL13161463 0.76 CENPE (0.69) CENPES1PR1S1PR5S1PR3XDH
SCHEMBL13184025 0.74 CENPE (0.40) CENPES1PR1MAPTTP53
SCHEMBL13161504 0.74 CENPE (0.68) CENPES1PR1S1PR5S1PR3XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742907-A4 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS INC (US) 2008-01-02 EP disclosed
EP-1742907-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2007-01-17 EP disclosed
WO-2005107762-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2005-11-17 WO disclosed