SCHEMBL4776165

SCHEMBL4776165

O=C(Cc1c[nH]c2ccccc12)Nc1cc(-c2cccnc2)nc(-c2ccccn2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 1/20 0.52
CDK4 P11802 1/20 0.52
CCND1 P24385 1/20 0.52
GLA P06280 1/20 0.48
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
MAPT P10636 3/20 0.46
ALDH1A1 P00352 1/20 0.46
PKM P14618 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 2/20 0.46
STAT3 P40763 2/20 0.46
HSD17B10 Q99714 1/20 0.46
EGFR P00533 1/20 0.44
ERBB2 P04626 1/20 0.44
POLB P06746 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769102 0.91 KMT2A (0.55) CDK4CCND1KMT2AMEN1MAPT
SCHEMBL2240341 0.87 CDK4 (0.50) CDK4CCND1KMT2AMEN1ALDH1A1
SCHEMBL3962080 0.83 CDK4 (0.58) CDK4CCND1KMT2AMEN1ALDH1A1
SCHEMBL4776020 0.82 CDK4 (0.49) CDK4CCND1KMT2AMEN1HTT
SCHEMBL4773415 0.82 ADORA2A (0.43) KMT2AMAPTALDH1A1CYP3A4CYP2C9
SCHEMBL4766487 0.81 CDK4 (0.47) CDK4CCND1KMT2AMEN1CDK2
SCHEMBL4766503 0.81 CDK4 (0.47) CDK4CCND1KMT2AMEN1CDK2
SCHEMBL4773620 0.81 CDK4 (0.47) CDK4CCND1KMT2AMEN1CDK2
SCHEMBL4768727 0.81 TDP1 (0.51) CDK4CCND1KMT2AMEN1MAPT
SCHEMBL4775038 0.81 CDK4 (0.47) CDK4CCND1KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed