SCHEMBL4769102

SCHEMBL4769102

O=C(CCc1c[nH]c2ccccc12)Nc1cc(-c2cccnc2)nc(-c2ccccn2)n1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.55
POLB P06746 2/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
CDK4 P11802 1/20 0.54
CCND1 P24385 1/20 0.54
MEN1 O00255 5/20 0.50
GBA1 P04062 1/20 0.46
MAPT P10636 4/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
SYK P43405 1/20 0.44
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GSK3B P49841 1/20 0.43
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776165 0.91 CCKBR (0.52) KMT2APOLBNPC1RAB9ACDK4
SCHEMBL3962080 0.85 CDK4 (0.58) KMT2APOLBNPC1RAB9ACDK4
SCHEMBL2240341 0.83 CDK4 (0.50) KMT2ANPC1RAB9ACDK4CCND1
SCHEMBL4766014 0.82 ADORA1 (0.47) POLBNPC1RAB9AGBA1ALDH1A1
SCHEMBL4771758 0.82 ADORA1 (0.43) KMT2APOLBNPC1RAB9AADORA3
SCHEMBL4770635 0.81 CYP1A2 (0.52) MAPTALDH1A1GAAADORA3ADORA2A
SCHEMBL4773065 0.81 ADORA1 (0.43) POLBNPC1RAB9AADORA3ADORA2A
SCHEMBL4776020 0.81 CDK4 (0.49) KMT2ACDK4CCND1MEN1GAA
SCHEMBL4768684 0.81 ADORA2A (0.43) KMT2AADORA3ADORA2AADORA1
SCHEMBL4765953 0.80 LMNA (0.52) NPC1RAB9AALDH1A1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed