SCHEMBL4776222

SCHEMBL4776222

CCCc1c(-c2ccc(OC)cc2F)cc(-c2ccc(OC)cc2)n1-c1ccc(OC)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
ALDH1A1 P00352 3/20 0.41
LMNA P02545 2/20 0.41
HTT P42858 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CHRNA7 P36544 2/20 0.37
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
ESR1 P03372 1/20 0.36
NPC1 O15118 1/20 0.35
MITF O75030 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
USP7 Q93009 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4779727 0.86 TP53 (0.41) TP53ALDH1A1LMNAHTTL3MBTL1
SCHEMBL4777615 0.81 CHRNA7 (0.42) TP53ALDH1A1LMNAHTTL3MBTL1
SCHEMBL4778456 0.81 ESR1 (0.56) LMNAESR1SMN1; SMN2USP7
SCHEMBL4778476 0.76 TP53 (0.43) TP53ALDH1A1LMNAHTTL3MBTL1
SCHEMBL4779710 0.71 TP53 (0.39) TP53ALDH1A1LMNAHTTL3MBTL1
SCHEMBL27781767 0.69 CYP2C19 (0.58) MEN1KMT2AKDM4ESMN1; SMN2USP7
SCHEMBL10340365 0.69 AMY1A (0.50) ALDH1A1MEN1HPGDKMT2ANPSR1
SCHEMBL21321935 0.68 APP (0.48) MAPTSMN1; SMN2
SCHEMBL19998337 0.67 MAOB (0.50) MAPT
SCHEMBL15694898 0.67 FLT3 (0.47) TP53ALDH1A1LMNAHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1889617-A1 Triphenyl modified 5-membered heterocycles and their use as anticancer and antiflammatory agents Freie Universität Berlin (DE) 2008-02-20 EP claimed
EP-1889617-A1 Triphenyl modified 5-membered heterocycles and their use as anticancer and antiflammatory agents Freie Universität Berlin (DE) 2008-02-20 EP disclosed
WO-2008006626-A1 TRIPHENYL MODIFIED 5-MEMBERED HETEROCYCLES AND THEIR USE AS ANTICANCER AND ANTIINFLAMMATORY AGENTS FREIE UNIVERSITÄT BERLIN (DE) 2008-01-17 WO disclosed