SCHEMBL4776570

SCHEMBL4776570

CC(C)Oc1cc(O)ccc1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
CA12 O43570 4/20 0.50
CA1 P00915 4/20 0.50
CA2 P00918 4/20 0.50
CA7 P43166 4/20 0.50
CA9 Q16790 4/20 0.50
CA14 Q9ULX7 4/20 0.50
TSHR P16473 1/20 0.50
ADRB3 P13945 7/20 0.49
ADRB1 P08588 6/20 0.49
ALOX5 P09917 1/20 0.46
PTGS2 P35354 1/20 0.46
IRAK4 Q9NWZ3 2/20 0.45
KDM4E B2RXH2 1/20 0.45
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6933447 0.88 ESR1 (0.51) ALDH1A1ESR1ESR2CA12CA1
SCHEMBL9774402 0.87 CA12 (0.50) ALDH1A1CA12CA1CA2CA7
SCHEMBL17908039 0.84 ALDH1A1 (0.73) ALDH1A1ADRB3ADRB1IRAK4KDM4E
SCHEMBL8235269 0.83 ESR1 (0.48) ALDH1A1ESR1ESR2CA12CA1
SCHEMBL711452 0.83 CA12 (0.59) ALDH1A1CA12CA1CA2CA7
SCHEMBL27051909 0.82 ESR1 (0.53) ALDH1A1ESR1ESR2CA12CA1
SCHEMBL1699147 0.82 ALDH1A1 (0.56) ALDH1A1ADRB3ADRB1IRAK4KDM4E
SCHEMBL27747073 0.82 ALDH1A1 (0.56) ALDH1A1CA12CA1CA2CA7
SCHEMBL25257928 0.81 ALDH1A1 (0.54) ALDH1A1ADRB3ADRB1IRAK4KDM4E
SCHEMBL6647244 0.81 ALDH1A1 (0.54) ALDH1A1CA1CA2TSHRADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1892239-B1 Inhibitors of cytosolic phospholipase A2 WYETH LLC (US) 2013-02-20 EP disclosed
EP-1892239-A1 Inhibitors of cytosolic phospholipase A2 Wyeth a Corporation of the State of Delaware (US) 2008-02-27 EP disclosed
EP-1451154-B1 INHIBITORS OF CYTOSOLIC PHOSPHOLIPASE A2 WYETH CORP (US) 2008-01-16 EP disclosed