SCHEMBL4777124

SCHEMBL4777124

CC(=O)N1CCC(C(=O)N(CCCN2CCC(Cc3ccccc3)CC2)Cc2ccc(Cl)c(Cl)c2)CC1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.67
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
GAA P10253 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5111655 0.95 CCR5 (0.63) CCR5
Trifluoroacetic Acid SCHEMBL4775617 0.86 CCR5 (0.64) CCR5
SCHEMBL4777105 0.86 CCR5 (0.84) CCR5
Trifluoroacetic Acid SCHEMBL4775779 0.86 CCR5 (0.64) CCR5KDM4ELMNAGAA
Trifluoroacetic Acid SCHEMBL4777069 0.85 CCR5 (0.68) CCR5KDM4ELMNAGAA
Trifluoroacetic Acid SCHEMBL4777927 0.84 CCR5 (0.64) CCR5KDM4ELMNAGAA
Trifluoroacetic Acid SCHEMBL4777815 0.83 CCR5 (0.63) CCR5KDM4ELMNAGAA
Trifluoroacetic Acid SCHEMBL4768574 0.83 CCR5 (0.63) CCR5KDM4ELMNAGAA
SCHEMBL7509134 0.81 CCR5 (0.70) CCR5KDM4ELMNAGAA
Trifluoroacetic Acid SCHEMBL4778140 0.81 CCR5 (0.60) CCR5KDM4ELMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1886994-A1 Cyclic amine compounds as CCR5 antagonists Takeda Pharmaceutical Company Limited (JP) 2008-02-13 EP disclosed