SCHEMBL4779112

SCHEMBL4779112

CS(=O)(=O)c1ccc(-c2cnc3nc(N)nc(N4CCOCC4)c3n2)cc1.Nc1nc(N2CCOCC2)c2nc(-c3ccc(C(F)(F)F)cc3)cnc2n1.Nc1nc(N2CCOCC2)c2nc(-c3ccc4[nH]ccc4c3)cnc2n1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.52
PIK3CA P42336 4/20 0.42
MTOR P42345 3/20 0.42
ATR Q13535 2/20 0.42
CYP2C9 P11712 1/20 0.42
PIK3CG P48736 1/20 0.41
MAP3K11 Q16584 1/20 0.41
AKT1 P31749 1/20 0.40
TGFBR1 P36897 1/20 0.40
PTGS2 P35354 1/20 0.38
GHSR Q92847 1/20 0.38
PRKDC P78527 1/20 0.38
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
GRIA1 P42261 1/20 0.37
KCNH2 Q12809 1/20 0.37
CHEK1 O14757 1/20 0.37
JAK2 O60674 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3755300 0.85 NOS1 (0.67) NOS1PIK3CAMTORATRCYP2C9
SCHEMBL4796117 0.84 NOS1 (0.51) NOS1PIK3CAMTORPIK3CGAKT1
SCHEMBL3760218 0.84 NOS1 (0.71) NOS1PIK3CAMTORATRPIK3CG
SCHEMBL3755502 0.82 NOS1 (0.74) NOS1PIK3CAMTORPIK3CGAKT1
SCHEMBL3760392 0.76 NOS1 (0.72) NOS1PIK3CAMTORPIK3CGJAK2
SCHEMBL3755637 0.76 NOS1 (0.72) NOS1PIK3CAMTORATRPIK3CG
SCHEMBL3765478 0.75 NOS1 (0.67) NOS1PIK3CAMTORAKT1
SCHEMBL3758149 0.75 NOS1 (0.74) NOS1PIK3CAMTORPIK3CGPRKDC
SCHEMBL3760949 0.74 NOS1 (0.69) NOS1PIK3CAMTORJAK2
SCHEMBL20985856 0.72 NOS1 (0.66) NOS1PIK3CAMTORATRPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009079-A2 SUBSTITUTED PTERIDINES USEFUL FOR THE TREATMENT AND PREVENTION OF VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed