SCHEMBL4780709

SCHEMBL4780709

CNC(=O)Cn1c(C(=O)N2CCOCC2)c(CN2CCC(c3c(F)cccc3Cl)CC2)c2ccccc21.Cc1c(CN2CCC(c3c(F)cccc3Cl)CC2)c2ccccc2n1CC(=O)N(C)C

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 2/20 0.37
POLB P06746 2/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CNR2 P34972 10/20 0.37
CNR1 P21554 2/20 0.37
CYP2A13 Q16696 1/20 0.35
MEN1 O00255 1/20 0.35
KRAS P01116 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRL1 P41146 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4779504 0.97 KMT2A (0.40) KMT2AKDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4779350 0.92 CYP2A13 (0.42) KMT2AKDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4780859 0.92 KMT2A (0.44) KMT2AKDM4EPOLBTSHRSMN1; SMN2
Hydrochloric Acid SCHEMBL4505962 0.86 OPRL1 (0.42) KMT2AKDM4EPOLBCNR2CNR1
SCHEMBL4774108 0.86 KDM4E (0.44) KMT2AKDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4778810 0.86 KDM4E (0.46) KMT2AKDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4706868 0.83 CYP2A13 (0.43) KMT2AKDM4EPOLBTSHRSMN1; SMN2
SCHEMBL4780556 0.83 KDM4E (0.46) KDM4EPOLBTSHRSMN1; SMN2CNR2
SCHEMBL4781123 0.82 CNR2 (0.48) KDM4ECNR2ALDH1A1TDP1OPRL1
SCHEMBL4780716 0.82 CNR1 (0.36) KMT2AKDM4EPOLBTSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008000818-A1 FLUORINATED INDOLEAMIDES USEFUL AS LIGANDS OF THE ORL-1 RECEPTOR BRANE DISCOVERY S.R.L. (IT) 2008-01-03 WO claimed