SCHEMBL4780962

SCHEMBL4780962

O=C(Nc1cccc2cnccc12)NC1C2CN(S(=O)(=O)c3ccccc3F)CC21

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
EPHX2 P34913 1/20 0.47
CNR1 P21554 1/20 0.46
TRPV1 Q8NER1 14/20 0.46
CHRM1 P11229 2/20 0.46
CYP3A4 P08684 2/20 0.45
P2RX7 Q99572 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778063 0.89 CHRM1 (0.48) EPHX2CNR1TRPV1CHRM1
SCHEMBL4781101 0.89 EPHX2 (0.51) KDM4EEPHX2CNR1TRPV1CHRM1
SCHEMBL4779491 0.87 TRPV1 (0.51) EPHX2TRPV1
SCHEMBL4779566 0.83 TRPV1 (0.50) EPHX2CNR1TRPV1
SCHEMBL4779435 0.83 EPHX2 (0.51) ALDH1A1EPHX2CNR1TRPV1CHRM1
SCHEMBL4778894 0.83 EPHX2 (0.49) EPHX2CNR1TRPV1CHRM1CYP3A4
SCHEMBL4780302 0.83 TRPV1 (0.52) KDM4EALDH1A1MAPTTRPV1CYP3A4
SCHEMBL4776335 0.82 TRPV1 (0.53) KDM4EALDH1A1MAPTEPHX2TRPV1
SCHEMBL4779427 0.82 EPHX2 (0.51) KDM4EALDH1A1MAPTEPHX2CNR1
SCHEMBL4774265 0.82 TRPV1 (0.52) EPHX2CNR1TRPV1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008010061-A2 3-AZABICYCLO [3.1.0] HEXANE VANILLOID RECEPTOR LIGANDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESSES FOR THEIR PREPARATION GLENMARK PHARMACEUTICALS S.A. (US) 2008-01-24 WO disclosed