SCHEMBL4783091

SCHEMBL4783091

Cc1ccc(C2c3cccn3CCCN2C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TP53 P04637 1/20 0.40
MAPT P10636 4/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
RHOC P08134 2/20 0.40
RHOA P61586 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TACR1 P25103 4/20 0.39
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4783999 0.91 KDM4E (0.50) ALDH1A1KDM4EL3MBTL1MAPTRHOC
SCHEMBL4784173 0.90 ALDH1A1 (0.39) ALDH1A1KDM4EL3MBTL1TP53MAPT
SCHEMBL4783442 0.86 MAPT (0.47) ALDH1A1KDM4EL3MBTL1TP53MAPT
SCHEMBL4781085 0.86 TACR1 (0.40) ALDH1A1KDM4EL3MBTL1RHOCRHOA
SCHEMBL4785528 0.73 TACR1 (0.46) RHOCRHOATACR1
SCHEMBL4781278 0.72 ALDH1A1 (0.38) ALDH1A1KDM4EL3MBTL1MAPTMEN1
SCHEMBL4048036 0.71 MAPT (0.43) ALDH1A1KDM4EL3MBTL1MAPTMEN1
SCHEMBL4781699 0.71 TACR1 (0.40) ALDH1A1RHOCRHOASMN1; SMN2TACR1
SCHEMBL4783584 0.71 TRPV1 (0.46) ALDH1A1KDM4EMAPTMEN1KMT2A
SCHEMBL4782716 0.71 TACR1 (0.40) ALDH1A1RHOCRHOASMN1; SMN2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008067222-A1 HETEROCYCLIC MODULATORS OF TGR5 KALYPSYS, INC. (US) 2008-06-05 WO disclosed
WO-2008067222-A1 HETEROCYCLIC MODULATORS OF TGR5 KALYPSYS, INC. (US) 2008-06-05 WO disclosed