SCHEMBL4783207

SCHEMBL4783207

CCOC(=O)c1cc(C#N)c(N2CCC(C(=O)OC(C)(C)C)CC2)nc1CC(=O)N1CCCC1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 13/20 0.45
ALDH1A1 P00352 7/20 0.44
KDM4E B2RXH2 5/20 0.44
L3MBTL1 Q9Y468 4/20 0.44
HPGD P15428 2/20 0.44
LMNA P02545 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAPT P10636 2/20 0.44
GAA P10253 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
CASP1 P29466 1/20 0.44
HTT P42858 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP2C9 P11712 5/20 0.44
CYP3A4 P08684 3/20 0.44
CHRM2 P08172 1/20 0.44
DRD3 P35462 1/20 0.44
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4172207 0.88 P2RY12 (0.46) P2RY12ALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL4166527 0.85 ALDH1A1 (0.47) P2RY12ALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL3208916 0.82 P2RY12 (0.62) P2RY12ALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL4786928 0.81 P2RY12 (0.44) P2RY12ALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL3226916 0.80 ALDH1A1 (0.55) P2RY12ALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL4180538 0.78 ALDH1A1 (0.41) P2RY12ALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL4164295 0.78 ALDH1A1 (0.40) P2RY12ALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL4183233 0.78 ALDH1A1 (0.43) P2RY12ALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL4179538 0.78 ALDH1A1 (0.40) P2RY12ALDH1A1KDM4EL3MBTL1HPGD
SCHEMBL4737215 0.78 ALDH1A1 (0.38) P2RY12ALDH1A1KDM4EL3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008085119-A1 NEW PYRIDINE ANALOGUES VIII 518 ASTRAZENECA AB (SE) 2008-07-17 WO disclosed