SCHEMBL4783343

SCHEMBL4783343

OCC1c2ccccc2CCN1c1nc(-c2cccc(O)c2)nc(N2CCC[C@H]2CO)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.41
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
IRAK4 Q9NWZ3 1/20 0.39
SYK P43405 2/20 0.38
MKNK1 Q9BUB5 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
PFKFB3 Q16875 1/20 0.37
IMPDH2 P12268 2/20 0.36
PIK3CA P42336 2/20 0.36
KRAS P01116 1/20 0.34
CCNE2 O96020 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
MTOR P42345 2/20 0.34
PDK2 Q15119 2/20 0.34
PDK4 Q16654 1/20 0.34
CDK1 P06493 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4784691 1.00 AOC3 (0.41) AOC3ESR1ESR2IRAK4SYK
SCHEMBL4784501 0.94 AOC3 (0.38) AOC3ESR1ESR2IRAK4SYK
SCHEMBL4784483 0.90 ESR1 (0.38) AOC3ESR1ESR2PFKFB3PIK3CA
SCHEMBL4784160 0.85 PIK3CA (0.42) ESR1ESR2PFKFB3PIK3CAMTOR
SCHEMBL4884094 0.85 PIK3CA (0.44) ESR1ESR2PFKFB3PIK3CAMTOR
SCHEMBL4785045 0.84 PIK3CA (0.39) ESR1ESR2PFKFB3PIK3CAMTOR
SCHEMBL4785055 0.84 PIK3CA (0.39) ESR1ESR2PFKFB3PIK3CAMTOR
SCHEMBL4785148 0.84 ESR1 (0.42) ESR1ESR2PFKFB3PIK3CAMTOR
SCHEMBL4784132 0.84 PIK3CA (0.44) ESR1ESR2PFKFB3PIK3CAMTOR
SCHEMBL4784088 0.83 PIK3CA (0.43) ESR1ESR2PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO claimed
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed