SCHEMBL4783554

SCHEMBL4783554

CCCCC1(CC)C(=O)[SH]c2cc(OCC(=O)N[C@@H](C(=O)NCCN)c3ccccc3)c(SC)cc2N(c2ccccc2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.43
ELANE P08246 1/20 0.35
GPR88 Q9GZN0 1/20 0.35
CTSD P07339 3/20 0.33
TACR1 P25103 1/20 0.32
TACR3 P29371 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5691316 0.94 NR1H4 (0.45) NR1H4ELANECTSD
SCHEMBL4741522 0.92 NR1H4 (0.44) NR1H4ELANECTSD
SCHEMBL5707135 0.92 NR1H4 (0.42) NR1H4ELANECTSD
SCHEMBL4662900 0.92 NR1H4 (0.42) NR1H4ELANECTSD
SCHEMBL4782192 0.92 NR1H4 (0.42) NR1H4ELANECTSD
SCHEMBL4729688 0.91 NR1H4 (0.43) NR1H4ELANECTSD
SCHEMBL5327298 0.91 NR1H4 (0.45) NR1H4ELANECTSD
SCHEMBL6629929 0.91 NR1H4 (0.45) NR1H4ELANECTSD
SCHEMBL3853019 0.90 NR1H4 (0.41) NR1H4ELANECTSD
SCHEMBL6527603 0.90 NR1H4 (0.45) NR1H4ELANECTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008039829-A2 DIPHENYLHETEROCYCLE CHOLESTEROL ABSORPTION INHIBITORS IRONWOOD PHARMACEUTICALS, INC. (US) 2008-04-03 WO disclosed