SCHEMBL4783587

SCHEMBL4783587

C[As](C)CCC(Oc1ccc(C(F)(F)F)cc1)c1ccc(C(=O)N2CCN(C3CCCCC3)CC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.56
SLC6A4 P31645 4/20 0.56
SLC6A2 P23975 1/20 0.47
SLC6A3 Q01959 1/20 0.47
CCR3 P51677 6/20 0.45
L3MBTL3 Q96JM7 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
KMT2A Q03164 1/20 0.43
ADRB2 P07550 1/20 0.43
KDM4E B2RXH2 3/20 0.43
POLB P06746 1/20 0.42
ALDH1A1 P00352 1/20 0.42
SCN9A Q15858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4783410 0.99 HRH3 (0.57) HRH3SLC6A4SLC6A2SLC6A3CCR3
SCHEMBL4921656 0.88 SLC6A4 (0.73) HRH3SLC6A4SLC6A2SLC6A3CCR3
SCHEMBL4921696 0.87 SLC6A4 (0.75) HRH3SLC6A4SLC6A2SLC6A3L3MBTL3
Trifluoroacetic Acid SCHEMBL4925697 0.84 SLC6A4 (0.70) HRH3SLC6A4SLC6A2SLC6A3L3MBTL3
SCHEMBL4784879 0.82 HRH3 (0.65) HRH3SLC6A4MEN1HPGDTSHR
SCHEMBL4918880 0.82 SLC6A4 (0.72) HRH3SLC6A4SLC6A2SLC6A3L3MBTL3
SCHEMBL4925879 0.72 HRH3 (1.00) HRH3SLC6A4
SCHEMBL4735283 0.72 HRH3 (1.00) HRH3SLC6A4
SCHEMBL4919787 0.71 SLC6A4 (0.59) HRH3SLC6A4SLC6A2CCR3
SCHEMBL4733830 0.71 HRH3 (0.83) HRH3SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064036-A1 SUBSTITUTED PHENYL PROPYL AMINES AS HISTAMINE H3 RECEPTOR AND SEROTONIN TRANSPORTER MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2008-05-29 WO claimed