SCHEMBL4784879

SCHEMBL4784879

CCC(C)N1CCN(C(=O)c2ccc(C(CC[As](C)C)Oc3ccc(C(F)(F)F)cc3)cc2)CC1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 6/20 0.65
SLC6A4 P31645 2/20 0.65
EPHX2 P34913 2/20 0.45
DRD3 P35462 2/20 0.42
HTR1A P08908 3/20 0.41
GPR183 P32249 1/20 0.41
SLC6A9 P48067 3/20 0.40
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
PRKAB2 O43741 1/20 0.39
PRKAG1 P54619 1/20 0.39
PRKAA2 P54646 1/20 0.39
PRKAA1 Q13131 1/20 0.39
PRKAG3 Q9UGI9 1/20 0.39
PRKAG2 Q9UGJ0 1/20 0.39
PRKAB1 Q9Y478 1/20 0.39
DRD2 P14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4919233 0.88 HRH3 (0.85) HRH3SLC6A4EPHX2SLC6A9
Trifluoroacetic Acid SCHEMBL4924383 0.84 HRH3 (0.79) HRH3SLC6A4SLC6A9
SCHEMBL4783410 0.83 HRH3 (0.57) HRH3SLC6A4GPR183MEN1HPGD
SCHEMBL4783587 0.82 HRH3 (0.56) HRH3SLC6A4MEN1HPGDTSHR
SCHEMBL4733830 0.79 HRH3 (0.83) HRH3SLC6A4SLC6A9
SCHEMBL4735283 0.79 HRH3 (1.00) HRH3SLC6A4EPHX2SLC6A9
SCHEMBL4925879 0.79 HRH3 (1.00) HRH3SLC6A4EPHX2SLC6A9
Trifluoroacetic Acid SCHEMBL4916696 0.77 HRH3 (0.78) HRH3SLC6A4SLC6A9
SCHEMBL4732424 0.73 SLC6A4 (0.75) HRH3SLC6A4HTR1ASLC6A9
SCHEMBL4921696 0.71 SLC6A4 (0.75) HRH3SLC6A4SLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008064036-A1 SUBSTITUTED PHENYL PROPYL AMINES AS HISTAMINE H3 RECEPTOR AND SEROTONIN TRANSPORTER MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2008-05-29 WO claimed