SCHEMBL4784983

SCHEMBL4784983

NC(=O)N(c1ccc(-c2cccc3[nH]nc(N)c23)cc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.62
KIT P10721 6/20 0.62
FLT3 P36888 6/20 0.62
ABL1 P00519 9/20 0.59
BCR P11274 6/20 0.59
LCK P06239 3/20 0.54
CSF1R P07333 3/20 0.54
FLT1 P17948 3/20 0.54
FYN P06241 2/20 0.54
LYN P07948 2/20 0.54
SRC P12931 2/20 0.54
FLT4 P35916 2/20 0.54
BLK P51451 2/20 0.54
EPHB4 P54760 2/20 0.53
TEK Q02763 2/20 0.53
DAPK3 O43293 1/20 0.50
PRKD3 O94806 1/20 0.50
MAP4K4 O95819 1/20 0.50
PAK4 O96013 1/20 0.50
NTRK1 P04629 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13372736 0.88 KDR (0.60) KDRKITFLT3ABL1BCR
SCHEMBL27636403 0.87 KDR (0.48) KDRKITFLT3ABL1BCR
SCHEMBL27657341 0.87 KDR (0.54) KDRKITFLT3ABL1BCR
SCHEMBL27657344 0.87 KDR (0.69) KDRKITFLT3ABL1BCR
SCHEMBL3363647 0.87 KDR (0.68) KDRKITFLT3ABL1BCR
SCHEMBL4784148 0.87 KDR (0.77) KDRKITFLT3ABL1BCR
SCHEMBL27657352 0.86 KDR (0.66) KDRKITFLT3ABL1BCR
SCHEMBL27636405 0.86 KDR (0.47) KDRKITFLT3ABL1BCR
SCHEMBL27657351 0.86 KDR (0.61) KDRKITFLT3ABL1BCR
SCHEMBL4739859 0.85 KDR (0.63) KDRKITFLT3ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN claimed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN claimed
CN-102417487-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB 2012-04-18 CN disclosed
CN-1826324-B indazole, Benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LABORATORIES (US) 2011-12-07 CN disclosed
CN-101827584-A Solid dispersion product of N-aryl ureido drugs ABBOTT GMBH & CO KG 2010-09-08 CN disclosed
WO-2008080110-A1 METHODS FOR TREATING MACULAR EDEMA AND PATHOLOGIC OCULAR ANGIOGENESIS USING A NEUROPROTECTIVE AGENT AND A RECEPTOR TYROSINE KINASE INHIBITOR ALCON, INC. (CH) 2008-07-03 WO disclosed
CN-1826324-A Indazole, benzisoxazole and benzisothiazole kinase inhibitors ABBOTT LAB (US) 2006-08-30 CN disclosed
US-20040235892-A1 Indazole and benzisoxazole kinase inhibitors ABBOTT LABORATORIES 2004-11-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040235892-A1 Indazole and benzisoxazole kinase inhibitors ABL1, MAP3K19, MAP3K1 KDR 800/4885KIT 238/4885FLT3 41/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.